SCHEMBL8008283

SCHEMBL8008283

CC(C)(C)[Si](C)(C)Oc1ccc(CCC(=O)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
MAPT P10636 1/20 0.46
CASP3 P42574 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HSD11B1 P28845 1/20 0.44
CES1 P23141 4/20 0.44
FAAH O00519 1/20 0.44
FFAR1 O14842 1/20 0.43
ABCB1 P08183 2/20 0.43
SRD5A2 P31213 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008498 0.86 RAB9A (0.50) NPC1RAB9AMAPTCASP3SENP8
SCHEMBL4266308 0.84 FFAR1 (0.53) FFAR1SRD5A2
SCHEMBL4000606 0.81 LMNA (0.48) NPC1RAB9AMAPT
SCHEMBL4211862 0.81 STS (0.52) NPC1RAB9AMAPTSRD5A2
SCHEMBL305427 0.81 TDP1 (0.50) MAPTTDP1FFAR1
SCHEMBL4261600 0.80 PREP (0.42) FFAR1
SCHEMBL8693803 0.80 KMT2A (0.51) NPC1RAB9AFFAR1
SCHEMBL8697433 0.80 NPSR1 (0.45) NPC1RAB9AMAPTCASP3SENP8
SCHEMBL2928400 0.79 NPC1 (0.87) NPC1RAB9AMAPTCASP3SENP8
SCHEMBL7535671 0.79 F2RL1 (0.46) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0935597-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1999-08-18 EP claimed
WO-1998019997-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1998-05-14 WO claimed
US-6046355-A TOLUENE-4-THIOSULFONIC ACID S-ESTERS AS CHEMICAL INTERMEDIATES FOR VIRICIDES AND ASPARTYL PROTEASE INHIBITORS; AIDS WARNER-LAMBERT COMPANY (US) 2000-04-04 US disclosed
EP-0935597-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1999-08-18 EP disclosed
WO-1998019997-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed