SCHEMBL8008735

SCHEMBL8008735

Cc1ccc(C(C)(C)C)c(SC2=C(O)CC(CCc3ccccc3)(c3ccc(OCCN4CCN(C(=O)OC(C)(C)C)CC4)cc3)OC2=O)c1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 3/20 0.37
GPR4 P46093 1/20 0.37
ACKR3 P25106 1/20 0.36
EPHX2 P34913 4/20 0.35
ADAM17 P78536 1/20 0.35
SIGMAR1 Q99720 3/20 0.35
ADORA3 P0DMS8 1/20 0.34
HTR2A P28223 1/20 0.34
HTR7 P34969 1/20 0.34
OPRM1 P35372 1/20 0.34
LTA4H P09960 1/20 0.34
HRH2 P25021 1/20 0.34
HRH1 P35367 1/20 0.34
GPR119 Q8TDV5 1/20 0.34
DRD3 P35462 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
DRD2 P14416 1/20 0.34
LDHA P00338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8010688 0.90 LTA4H (0.39) LTA4HALDH1A1LDHA
SCHEMBL8008687 0.85 LDHA (0.41) LDHA
SCHEMBL8007680 0.82 LDHA (0.37) LDHA
SCHEMBL8014088 0.76 LTA4H (0.34) LTA4HALDH1A1LDHA
SCHEMBL8010546 0.76 LDHA (0.40) LDHA
SCHEMBL8010782 0.72 LDHA (0.38) ADORA3HTR2ALDHA
SCHEMBL7444083 0.72 LTA4H (0.48) EPHX2LTA4HALDH1A1
SCHEMBL8011472 0.69 LDHA (0.47) LDHA
SCHEMBL6604343 0.69 LDHA (0.48) LDHA
SCHEMBL14453585 0.69 KCNA5 (0.62) KCNA5GPR4EPHX2HRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046355-A TOLUENE-4-THIOSULFONIC ACID S-ESTERS AS CHEMICAL INTERMEDIATES FOR VIRICIDES AND ASPARTYL PROTEASE INHIBITORS; AIDS WARNER-LAMBERT COMPANY (US) 2000-04-04 US disclosed
EP-0935597-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1999-08-18 EP disclosed
WO-1998019997-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed