SCHEMBL8010647

SCHEMBL8010647

CCNS(=O)(=O)c1ccc(Oc2ccc(Br)c(C=O)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 1/20 0.43
CYP2C9 P11712 1/20 0.41
MMP1 P03956 3/20 0.41
ADAMTS4 O75173 2/20 0.41
MMP2 P08253 2/20 0.41
MMP13 P45452 2/20 0.41
MMP14 P50281 2/20 0.41
ADAMTS5 Q9UNA0 2/20 0.41
MEP1B Q16820 1/20 0.41
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862828 0.83 ALDH1A1 (0.43) ALDH1A1LMNASMN1; SMN2HTTMMP1
SCHEMBL7857418 0.80 HTT (0.42) ALDH1A1LMNASMN1; SMN2HTTMAPT
SCHEMBL7857250 0.79 SMN1; SMN2 (0.66) ALDH1A1LMNASMN1; SMN2HTTMAPT
SCHEMBL20157457 0.77 ALDH1A1 (0.56) ALDH1A1LMNASMN1; SMN2CYP2C9PKM
SCHEMBL7862803 0.77 HTT (0.39) ALDH1A1LMNASMN1; SMN2HTTMMP1
SCHEMBL29746806 0.75 HTT (0.44) ALDH1A1LMNASMN1; SMN2HTTCYP2C9
SCHEMBL7865553 0.75 ALDH1A1 (0.51) ALDH1A1LMNAHTTCYP2C9MAPT
SCHEMBL7863855 0.75 HTT (0.44) ALDH1A1LMNASMN1; SMN2HTTCYP2C9
SCHEMBL19622354 0.75 LMNA (0.37) ALDH1A1LMNASMN1; SMN2HTTCYP2C9
SCHEMBL14748381 0.74 ALDH1A1 (0.37) ALDH1A1LMNASMN1; SMN2HTTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2564857-A1 Boron-containing small molecules as anti-inflammatory agents Anacor Pharmaceuticals, Inc. (US) 2013-03-06 EP disclosed
WO-2009111676-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS ANACOR PHARMACEUTICALS, INC (US) 2009-09-11 WO disclosed