SCHEMBL8012121

SCHEMBL8012121

CC(=O)N1C(=O)C(=C(O)c2ccc(C(F)(F)F)cc2)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 3/20 0.42
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
PHGDH O43175 1/20 0.39
CASP1 P29466 2/20 0.39
CASP3 P42574 2/20 0.39
CASP4 P49662 2/20 0.39
CASP7 P55210 2/20 0.39
CASP9 P55211 2/20 0.39
CASP6 P55212 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
PAX8 Q06710 1/20 0.39
SLC6A9 P48067 1/20 0.38
SLC6A5 Q9Y345 1/20 0.38
NR1H2 P55055 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8012118 1.00 SNCA (0.42) SNCACA12CA9PHGDHCASP1
SCHEMBL8009610 0.87 CA12 (0.46) SNCACA12CA9CASP1CASP3
SCHEMBL8009607 0.87 CA12 (0.46) SNCACA12CA9CASP1CASP3
SCHEMBL8010160 0.86 MEN1 (0.44) SNCACA12CA9CASP1CASP3
SCHEMBL28408693 0.86 ALDH1A1 (0.44) SNCACA12CA9CASP1CASP3
SCHEMBL8010164 0.86 MEN1 (0.44) SNCACA12CA9CASP1CASP3
SCHEMBL4306349 0.85 AKR1C3 (0.41) MAPTSLC6A9SLC6A5NR1H2NR1H3
SCHEMBL4306346 0.85 AKR1C3 (0.41) MAPTSLC6A9SLC6A5NR1H2NR1H3
SCHEMBL4300692 0.84 MAPK1 (0.48) SNCACA12CA9KDM4EMAPT
SCHEMBL4300695 0.84 MAPK1 (0.48) SNCACA12CA9KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed