SCHEMBL8014606

SCHEMBL8014606

COc1cccc(-c2ccc3c(c2)CC[C@@H](CN(C)C)C3=O)c1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 4/20 0.59
THRA P10827 1/20 0.55
THRB P10828 1/20 0.55
HSP90AA1 P07900 1/20 0.55
CCR6 P51684 1/20 0.55
CYP24A1 Q07973 6/20 0.53
CYP27A1 Q02318 3/20 0.53
CYP26A1 O43174 4/20 0.52
CYP19A1 P11511 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7592165 1.00 METAP1 (0.59) METAP1THRATHRBHSP90AA1CCR6
SCHEMBL28031701 0.87 CYP26A1 (0.57) METAP1THRATHRBCYP24A1CYP27A1
SCHEMBL8012038 0.86 METAP1 (0.78) METAP1THRATHRBHSP90AA1CCR6
SCHEMBL7590283 0.86 METAP1 (0.78) METAP1THRATHRBHSP90AA1CCR6
Hydrochloric Acid SCHEMBL10341505 0.85 METAP1 (0.78) METAP1THRATHRBHSP90AA1CCR6
SCHEMBL7590969 0.79 METAP1 (0.74) METAP1THRATHRBHSP90AA1CCR6
SCHEMBL11011369 0.79 METAP1 (0.76) METAP1THRATHRBHSP90AA1CCR6
Hydrochloric Acid SCHEMBL4623159 0.78 METAP1 (0.78) METAP1THRATHRBHSP90AA1CCR6
SCHEMBL2969421 0.77 HSP90AA1 (0.55) METAP1HSP90AA1CCR6
Hydrochloric Acid SCHEMBL6293297 0.76 HSP90AA1 (0.57) METAP1HSP90AA1CCR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022895-A Substituted amino compounds and their use as substances having an analgesic effect GRUENENTHAL GMBH (DE) 2000-02-08 US disclosed