SCHEMBL8015200

SCHEMBL8015200

CC(=O)C(=Cc1cccc(C#N)c1Cl)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
KMT2A Q03164 3/20 0.34
LMNA P02545 2/20 0.34
PKM P14618 1/20 0.34
NOTUM Q6P988 1/20 0.34
CRHR1 P34998 3/20 0.34
XDH P47989 1/20 0.33
AKR1C3 P42330 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA7 P43166 1/20 0.33
APEX1 P27695 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL819819 0.80 KMT2A (0.44) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL822890 0.80 KMT2A (0.44) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8487129 0.80 NOTUM (0.34) KDM4EKMT2ANOTUMCRHR1XDH
SCHEMBL8018607 0.79 LMNA (0.45) KDM4EKMT2ALMNAPKMMEN1
SCHEMBL8018603 0.79 LMNA (0.45) KDM4EKMT2ALMNAPKMMEN1
SCHEMBL11862771 0.77 CYP1A2 (0.44) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL20954588 0.75 KDM4E (0.37) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL22400535 0.75 KDM4E (0.37) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9477461 0.73 CA1 (0.52) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9477455 0.73 CA1 (0.52) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36607-E Pyrrolidine compounds and process of preparing BAYER AKTIENGESELLSCHAFT (DE) 2000-03-07 US disclosed
US-5910593-A Highly selective process for the preparation of enantiomerically pure phenylsubstituted 1,4-dihydropyridine-3,5-dicarboxylic acid derivatives BAYER AKTIENGESELLSCHAFT (DE) 1999-06-08 US disclosed
US-5849924-A Highly selective process for the preparation of enantiomerically pure phenyl-substituted 1,4-dihydropyridine-3,5-dicarboxylic acid derivatives BAYER AKTIENGESELLSCAHFT (DE) 1998-12-15 US disclosed
US-5700948-A CALCIUM ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 1997-12-23 US disclosed