SCHEMBL8487129

SCHEMBL8487129

CC(=O)/C(C=O)=C/c1cccc(C#N)c1Cl

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.34
CRHR1 P34998 3/20 0.34
P2RX7 Q99572 4/20 0.33
KMT2A Q03164 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 3/20 0.32
GAA P10253 3/20 0.32
CASP3 P42574 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
XDH P47989 1/20 0.31
TRPA1 O75762 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GLA P06280 1/20 0.31
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537617 0.80 KMT2A (0.44) KMT2AL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL4537616 0.80 KMT2A (0.44) KMT2AL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8015200 0.80 KDM4E (0.38) NOTUMCRHR1KMT2AL3MBTL1KDM4E
SCHEMBL2895077 0.74 MEN1 (0.41) KMT2AKDM4EALDH1A1GAACASP3
SCHEMBL30783064 0.74 MEN1 (0.41) KMT2AKDM4EALDH1A1GAACASP3
SCHEMBL8018603 0.71 LMNA (0.45) KMT2AL3MBTL1KDM4EALDH1A1GAA
SCHEMBL8018607 0.71 LMNA (0.45) KMT2AL3MBTL1KDM4EALDH1A1GAA
SCHEMBL16953233 0.71 TRPA1 (0.36) KDM4EALDH1A1GAACASP3SENP8
SCHEMBL31251566 0.70 SMN1; SMN2 (0.38) KMT2AL3MBTL1ALDH1A1GAATRPA1
SCHEMBL15547200 0.70 CA1 (0.46) KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0716081-B1 Highly selective process for the preparation of enantiomerically pure phenyl-substituted 1,4-dihydropyridine-3,5-dicarboxylic acid derivatives BAYER HEALTHCARE AG (DE) 2006-04-05 EP disclosed