SCHEMBL8017165

SCHEMBL8017165

CC(=O)N1C(=O)/C(=C(/Cl)c2ccc(Br)cc2)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 1/20 0.43
PAX8 Q06710 1/20 0.43
MAPT P10636 2/20 0.41
SNCA P37840 3/20 0.41
CASP1 P29466 2/20 0.41
CASP3 P42574 2/20 0.41
CASP4 P49662 2/20 0.41
CASP7 P55210 2/20 0.41
CASP9 P55211 2/20 0.41
CASP6 P55212 2/20 0.41
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8017167 1.00 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ALMNACYP1A2
SCHEMBL6325583 0.93 CASP1 (0.44) ALDH1A1LMNAMAPTSNCACASP1
SCHEMBL6325589 0.93 CASP1 (0.44) ALDH1A1LMNAMAPTSNCACASP1
SCHEMBL6328679 0.90 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL6328682 0.90 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL6321810 0.90 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ALMNAPAX8
SCHEMBL6321814 0.90 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ALMNAPAX8
SCHEMBL8010160 0.88 MEN1 (0.44) ALDH1A1MEN1KMT2ALMNACYP1A2
SCHEMBL8010164 0.88 MEN1 (0.44) ALDH1A1MEN1KMT2ALMNACYP1A2
SCHEMBL6327330 0.87 SNCA (0.52) ALDH1A1MEN1KMT2ALMNAPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed