SCHEMBL8017351

SCHEMBL8017351

C1=C(c2c[nH]c3ncccc23)CCNC1.c1cnc2[nH]ccc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.51
DRD2 P14416 2/20 0.51
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.51
ALOX15 P16050 1/20 0.51
HSD17B10 Q99714 1/20 0.51
AXL P30530 1/20 0.49
NUDT1 P36639 1/20 0.49
HTR2A P28223 2/20 0.45
HTR2B P41595 1/20 0.45
IKBKE Q14164 1/20 0.43
TBK1 Q9UHD2 1/20 0.43
TMEM97 Q5BJF2 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
DYRK1A Q13627 2/20 0.42
HTR1A P08908 2/20 0.42
ADRA1D P25100 1/20 0.42
SLC6A4 P31645 1/20 0.42
ADRA1A P35348 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1848853 0.90 HTR2C (0.61) HTR2CDRD2KDM4EALDH1A1MAPT
SCHEMBL10124857 0.79 CDK9 (0.49) HTR2CDRD2KDM4EALDH1A1MAPT
SCHEMBL12874727 0.74 HTR2C (0.51) HTR2CDRD2KDM4EALDH1A1MAPT
SCHEMBL3930943 0.73 DYRK1A (0.42) HTR2CAXLNUDT1HTR2AHTR2B
SCHEMBL12874723 0.73 HTR2C (0.46) HTR2CDRD2KDM4EALDH1A1MAPT
SCHEMBL24440670 0.72 HTR2A (0.57) HTR2CAXLHTR2AHTR2BIKBKE
Piperazine SCHEMBL27563143 0.72 NUDT1 (0.81) HTR2CAXLNUDT1HTR2ASLC6A4
SCHEMBL38661232 0.72 HTR2C (0.49) HTR2CDRD2KDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL27893779 0.71 AXL (0.95) KDM4EALDH1A1MAPTALOX15AXL
Hydrochloric Acid SCHEMBL5325493 0.71 AXL (0.95) KDM4EALDH1A1MAPTALOX15AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000040581-A1 3,4-DIHYDRO-2H-BENZO[1,4]OXAZINE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-07-13 WO disclosed