SCHEMBL8018940

SCHEMBL8018940

CSc1ccc(C(O)C#N)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.54
ALOX5 P09917 4/20 0.47
SLC6A4 P31645 3/20 0.42
ACACB O00763 1/20 0.39
AKR1C3 P42330 3/20 0.36
AKR1C2 P52895 3/20 0.36
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PLK1 P53350 1/20 0.34
MAOA P21397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2195029 0.79 ALOX5 (0.43) ALOX5SLC6A4ACACBAKR1C3AKR1C2
SCHEMBL3991740 0.76 TSHR (0.60) TSHRALOX5ESR1ESR2ALDH1A1
SCHEMBL8019231 0.76 TSHR (0.60) TSHRALOX5ESR1ESR2ALDH1A1
SCHEMBL1200882 0.76 TSHR (0.60) TSHRALOX5ESR1ESR2ALDH1A1
SCHEMBL15775527 0.75 SLC6A4 (0.57) ALOX5SLC6A4ACACBNOS3NOS1
SCHEMBL6182478 0.75 SLC6A4 (0.50) ALOX5SLC6A4ACACBAKR1C3AKR1C2
SCHEMBL13557508 0.75 SLC6A4 (0.50) ALOX5SLC6A4ACACBAKR1C3AKR1C2
SCHEMBL11811969 0.75 ACACB (0.43) ALOX5SLC6A4ACACBAKR1C3AKR1C2
Hydrochloric Acid SCHEMBL15775544 0.73 SLC6A4 (0.55) ALOX5SLC6A4ACACBNOS3NOS1
SCHEMBL2197891 0.73 ALOX5 (0.46) ALOX5SLC6A4ACACBAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610048-B1 Process for producing optically active alpha-hydrocarboxylic acid having phenyl group MITSUBISHI RAYON CO (JP) 1999-09-22 EP claimed
US-5580765-A A CULTURE PRODUCT OF A-HYDROXYNITRILE OR A MIXTURE OF ALDEHYDE AND PRUSSIC ACID NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1996-12-03 US claimed
EP-0610048-A2 Process for producing optically active alpha-hydrocarboxylic acid having phenyl group NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1994-08-10 EP claimed
EP-0711836-B1 Method of producing optically active alpha-hydroxy acid or alpha-hydroxyamide MITSUBISHI RAYON CO (JP) 2000-02-02 EP disclosed
EP-0610048-B1 Process for producing optically active alpha-hydrocarboxylic acid having phenyl group MITSUBISHI RAYON CO (JP) 1999-09-22 EP disclosed
US-5736385-A NITRILASE OR NITRILE HYDRATASE HYDROLYSIS OF A CYANOHYDRIN WHILE AUTOMATICALLY CONTROLLING CYANOHYDRIN CONCENTRATION NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1998-04-07 US disclosed
US-5580765-A A CULTURE PRODUCT OF A-HYDROXYNITRILE OR A MIXTURE OF ALDEHYDE AND PRUSSIC ACID NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1996-12-03 US disclosed
EP-0711836-A1 Method of producing optically active alpha-hydroxy acid or alpha-hydroxyamide NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1996-05-15 EP disclosed
EP-0610048-A2 Process for producing optically active alpha-hydrocarboxylic acid having phenyl group NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1994-08-10 EP disclosed