SCHEMBL8019368

SCHEMBL8019368

NC(=O)CCc1csc2ccc(OCc3ccccc3)cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 4/20 0.53
MTNR1A P48039 3/20 0.46
TNKS2 Q9H2K2 1/20 0.46
PARP2 Q9UGN5 1/20 0.46
EDNRA P25101 1/20 0.45
PARP10 Q53GL7 1/20 0.45
FFAR4 Q5NUL3 1/20 0.44
MTNR1B P49286 2/20 0.44
PPARG P37231 2/20 0.44
PPARD Q03181 2/20 0.44
PPARA Q07869 2/20 0.44
PLAU P00749 1/20 0.43
PLAT P00750 1/20 0.43
SPHK2 Q9NRA0 1/20 0.43
SPHK1 Q9NYA1 1/20 0.43
MEN1 O00255 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
LTA4H P09960 1/20 0.43
PLA2G2A P14555 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8694064 0.91 PPARD (0.53) FFAR1TNKS2PARP2PARP10FFAR4
SCHEMBL8695196 0.91 FFAR1 (0.64) FFAR1MTNR1AEDNRAFFAR4PPARG
SCHEMBL8695194 0.81 PPARD (0.58) FFAR1FFAR4PPARGPPARDPPARA
SCHEMBL3882956 0.79 MAOB (0.56) FFAR1PARP10FFAR4SPHK2SPHK1
SCHEMBL30656241 0.78 FFAR1 (0.56) FFAR1TNKS2PARP2EDNRAFFAR4
SCHEMBL8694056 0.75 F9 (0.50) FFAR1EDNRAPARP10FFAR4SPHK2
SCHEMBL30138881 0.75 CYP2A6 (0.58) MTNR1A
SCHEMBL8905373 0.75 CYP2A6 (0.58) MTNR1A
SCHEMBL6234342 0.74 MAOB (0.51) FFAR1TNKS2PARP2EDNRA
SCHEMBL2912575 0.74 FFAR1 (0.66) FFAR1PARP10FFAR4SPHK2SPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745584-B1 Arylalkyl(thio) carboxamides compounds with affinity for melatonine receptors, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-01-05 EP disclosed
US-5721276-A TREATING DISORDERS OF MELATONINERGIC SYSTEM ADIR ET COMPAGNIE (FR) 1998-02-24 US disclosed
EP-0745584-A1 Arylalkyl(thio) carboxamides compounds with affinity for melatonine receptors, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-12-04 EP disclosed