SCHEMBL8019454

SCHEMBL8019454

O=C1Cc2ccccc2C(=O)N1CCCCCCCCCC(O)CO

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.53
MAPT P10636 4/20 0.53
APAF1 O14727 3/20 0.53
ALDH1A1 P00352 3/20 0.53
GAA P10253 3/20 0.53
BLM P54132 2/20 0.53
CASP1 P29466 1/20 0.53
RAB9A P51151 1/20 0.53
CASP7 P55210 1/20 0.53
HSD17B10 Q99714 1/20 0.53
MEN1 O00255 4/20 0.49
HPGD P15428 2/20 0.49
HDAC8 Q9BY41 4/20 0.47
HDAC1 Q13547 4/20 0.47
HDAC7 Q8WUI4 4/20 0.47
HDAC3 O15379 3/20 0.47
HDAC4 P56524 3/20 0.47
HDAC2 Q92769 3/20 0.47
HDAC10 Q969S8 3/20 0.47
HDAC11 Q96DB2 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8070540 0.84 KMT2A (0.61) KMT2AMAPTAPAF1ALDH1A1GAA
SCHEMBL6779279 0.84 TDP1 (0.54) KMT2AALDH1A1MEN1HPGDHDAC8
SCHEMBL6778346 0.84 TDP1 (0.54) KMT2AALDH1A1MEN1HPGDHDAC8
SCHEMBL20707259 0.82 HDAC1 (0.53) KMT2AMAPTALDH1A1RAB9AMEN1
SCHEMBL6774135 0.82 HDAC1 (0.53) KMT2AMAPTALDH1A1RAB9AMEN1
SCHEMBL11283988 0.81 KMT2A (0.64) KMT2AMAPTAPAF1ALDH1A1GAA
SCHEMBL8375889 0.81 KMT2A (0.44) KMT2AMAPTAPAF1ALDH1A1GAA
SCHEMBL11852813 0.79 KMT2A (0.61) KMT2AMAPTAPAF1ALDH1A1GAA
SCHEMBL11280189 0.78 KMT2A (0.68) KMT2AMAPTAPAF1ALDH1A1GAA
SCHEMBL751414 0.78 ALDH1A1 (0.54) MAPTALDH1A1RAB9AHDAC8HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6133274-A TREATING DISEASE MEDIATED BY INTRACELLULAR SIGNALING THROUGH ONE OR TWO SPECIFIC INTRACELLULAR SIGNALING PATHWAYS; A XANTHINYL HAVING AT LEAST ONE NITROGEN SUBSTITUTED BY AN HYDROXYALKYL; ANTITUMOR,-CARCINOGENIC,-ARTHRITIC AGENTS CELL THERAPEUTICS, INC. (US) 2000-10-17 US disclosed