SCHEMBL8019526

SCHEMBL8019526

CN1CCN(c2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccccc23)CC1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.65
HTR6 P50406 4/20 0.62
POLB P06746 3/20 0.62
ALDH1A1 P00352 2/20 0.61
HPGD P15428 2/20 0.61
CRHBP P24387 2/20 0.61
CRHR2 Q13324 2/20 0.61
MAPT P10636 1/20 0.61
LMNA P02545 1/20 0.60
TP53 P04637 2/20 0.60
RXFP1 Q9HBX9 2/20 0.58
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8019523 0.91 HTR6 (0.70) THRBHTR6POLBALDH1A1HPGD
SCHEMBL8029242 0.89 CRHBP (0.74) THRBHTR6POLBALDH1A1HPGD
SCHEMBL8027278 0.85 HTR6 (0.85) THRBHTR6POLBMAPTRXFP1
SCHEMBL8029081 0.80 HPGD (0.84) THRBHTR6POLBALDH1A1HPGD
SCHEMBL8028196 0.80 HPGD (0.84) THRBHTR6POLBALDH1A1HPGD
SCHEMBL8019460 0.79 HTR6 (0.60) THRBHTR6ALDH1A1HPGDMAPT
SCHEMBL8026556 0.79 KDM4E (0.64) THRBHTR6POLBALDH1A1HPGD
SCHEMBL8019326 0.77 HTR6 (0.98) THRBHTR6POLBMAPTRXFP1
SCHEMBL8030163 0.75 HTR6 (1.00) HTR6POLBMAPTRXFP1
SCHEMBL8019071 0.75 HTR6 (0.76) HTR6POLBMAPTLMNARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed