SCHEMBL8019647

SCHEMBL8019647

CCOC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)c1ccc(Cl)c(NC(NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.45
CTSS P25774 3/20 0.44
ACE P12821 1/20 0.44
CTSL P07711 2/20 0.43
GPR139 Q6DWJ6 1/20 0.43
CTSB P07858 1/20 0.43
CTSK P43235 1/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6773066 0.84 CTSS (0.44) KLK5CTSSGPR139RAB9ANPC1
SCHEMBL8009085 0.84 GPR139 (0.46) CTSSGPR139RAB9ANPC1MAPT
SCHEMBL6773596 0.81 GPR139 (0.51) CTSSGPR139RAB9ATP53
SCHEMBL1673615 0.81 KLK5 (0.56) KLK5CTSSACECTSLCTSB
SCHEMBL1673614 0.81 KLK5 (0.56) KLK5CTSSACECTSLCTSB
SCHEMBL12122453 0.76 CTSS (0.64) KLK5CTSSACECTSLCTSB
SCHEMBL1273042 0.76 CTSS (0.64) KLK5CTSSACECTSLCTSB
SCHEMBL26818324 0.74 CTSS (0.49) KLK5CTSSACECTSLCTSB
SCHEMBL23332639 0.73 KLK5 (0.59) KLK5CTSSACECTSLCTSB
SCHEMBL28582380 0.73 KLK5 (0.59) KLK5CTSSACECTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028223-A AN INTEGRIN ANTAGONISTS TREATING BONE DISORDER, PERIODONTAL DISEASE, OSTEOPOROSIS, HUMORAL HYPERCALCEMIA OF MALIGNANCY, PAGET'S DISEASE, TUMOR ANGIOGENESIS, DIABETIC RETINOPATHY, ARTHRITIS, SMOOTH MUSCLE CELL MIGRATION AND RESTENOSIS G. D. SEARLE & CO. (US) 2000-02-22 US disclosed