SCHEMBL8020973

SCHEMBL8020973

CC(C)(C)c1ccccc1C1=C[C@@]2(C)[C@@H](CC[C@H]3[C@@H]4CCC[C@@]4(C)CC[C@@H]32)NC1=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 3/20 0.41
SRD5A1 P18405 9/20 0.35
CYP19A1 P11511 3/20 0.34
SRD5A2 P31213 7/20 0.33
LMNA P02545 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
ABCC4 O15439 1/20 0.33
ABCB11 O95342 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CHRM1 P11229 1/20 0.33
HSD3B1 P14060 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33
THPO P40225 1/20 0.33
BLM P54132 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8016925 0.86 MBOAT4 (0.43) MBOAT4SRD5A1CYP19A1SRD5A2
SCHEMBL8023955 0.82 MBOAT4 (0.45) MBOAT4SRD5A1CYP19A1SRD5A2LMNA
SCHEMBL8006675 0.81 MBOAT4 (0.41) MBOAT4SRD5A1CYP19A1SRD5A2LMNA
SCHEMBL8016784 0.78 MBOAT4 (0.42) MBOAT4SRD5A1CYP19A1SRD5A2
SCHEMBL5109022 0.77 MBOAT4 (0.51) MBOAT4SRD5A1CYP19A1SRD5A2LMNA
SCHEMBL8023129 0.77 MBOAT4 (0.45) MBOAT4SRD5A1CYP19A1SRD5A2LMNA
SCHEMBL8020270 0.76 SRD5A1 (0.42) MBOAT4SRD5A1CYP19A1SRD5A2LMNA
SCHEMBL9618180 0.74 SRD5A1 (0.44) MBOAT4SRD5A1SRD5A2
SCHEMBL8407145 0.73 MBOAT4 (0.47) MBOAT4SRD5A1CYP19A1
SCHEMBL8020709 0.73 MBOAT4 (0.35) MBOAT4SRD5A1CYP19A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP claimed