SCHEMBL8021409

SCHEMBL8021409

COC(=O)c1ccccc1C(c1ccccc1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
ALDH1A1 P00352 3/20 0.53
TDP1 Q9NUW8 3/20 0.53
GAA P10253 2/20 0.53
TSHR P16473 3/20 0.52
LMNA P02545 1/20 0.52
CFTR P13569 1/20 0.50
HSD17B10 Q99714 1/20 0.50
KDM4E B2RXH2 2/20 0.49
ATM Q13315 2/20 0.49
MAPT P10636 1/20 0.49
ALOX15 P16050 1/20 0.49
POLB P06746 1/20 0.49
SLC6A3 Q01959 1/20 0.47
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA5A P35218 1/20 0.45
CA9 Q16790 1/20 0.45
MYC P01106 1/20 0.44
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7186547 0.84 ALDH1A1 (0.45) KMT2AALDH1A1TDP1GAATSHR
SCHEMBL4068453 0.84 TSHR (0.50) KMT2AALDH1A1TDP1GAATSHR
Hydrogen Peroxide SCHEMBL28473316 0.83 TSHR (0.57) KMT2AALDH1A1TDP1GAATSHR
SCHEMBL11274330 0.83 TSHR (0.49) KMT2AALDH1A1TDP1GAATSHR
SCHEMBL11030148 0.83 TSHR (0.49) KMT2AALDH1A1TDP1GAATSHR
SCHEMBL28323865 0.81 TSHR (0.47) KMT2AALDH1A1TDP1GAATSHR
SCHEMBL9305621 0.81 KDM4E (0.53) KMT2AALDH1A1TDP1GAATSHR
SCHEMBL254882 0.81 TSHR (0.59) KMT2AALDH1A1TDP1GAATSHR
SCHEMBL996468 0.79 TSHR (0.57) KMT2AALDH1A1GAATSHRLMNA
SCHEMBL8945914 0.79 ALDH1A1 (0.79) KMT2AALDH1A1TDP1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000030632-A1 ARYL AND HETEROARYL COMPOUNDS USEFUL AS FIBROBLAST GROWTH FACTOR ANTAGONISTS EISAI CO., LTD. (JP) 2000-06-02 WO claimed
CN-105237560-B A kind of LZC696 intermediates and its synthetic method 上海博氏医药科技有限公司 2018-07-06 CN disclosed
US-7531573-B2 potent, selective and safe inhibitors of the Ca2+-activated potassium channel CHILDREN'S MEDICAL CENTER CORPORATION (US) 2009-05-12 US disclosed
US-7531573-B2 potent, selective and safe inhibitors of the Ca2+-activated potassium channel CHILDREN'S MEDICAL CENTER CORPORATION (US) 2009-05-12 US disclosed
WO-2000030632-A1 ARYL AND HETEROARYL COMPOUNDS USEFUL AS FIBROBLAST GROWTH FACTOR ANTAGONISTS EISAI CO., LTD. (JP) 2000-06-02 WO disclosed