SCHEMBL8021729

SCHEMBL8021729

C=CCc1ccc2cccc(CCCN)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.40
MTNR1A P48039 5/20 0.39
MTNR1B P49286 2/20 0.39
TLR8 Q9NR97 4/20 0.39
SSTR2 P30874 2/20 0.37
SSTR4 P31391 2/20 0.37
XDH P47989 1/20 0.36
CYP1A2 P05177 2/20 0.36
MAPT P10636 2/20 0.36
MC4R P32245 1/20 0.36
MC5R P33032 1/20 0.36
MC3R P41968 1/20 0.36
MC1R Q01726 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
GPR84 Q9NQS5 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033335 0.81 TLR8 (0.47) MTNR1ATLR8SSTR2SSTR4CYP1A2
SCHEMBL8021660 0.79 TLR8 (0.49) MTNR1ATLR8CYP1A2CYP2D6CYP2C19
SCHEMBL8031004 0.78 TLR8 (0.51) MTNR1ATLR8CYP1A2CYP2D6CYP2C19
SCHEMBL8034939 0.77 TLR8 (0.56) TLR8
SCHEMBL8021705 0.76 TLR8 (0.55) TLR8
SCHEMBL8033115 0.74 CYP2A6 (0.50) NQO2MTNR1AMTNR1BTLR8SSTR2
SCHEMBL10344605 0.73 S1PR1 (0.43) TLR8CNR1CNR2
SCHEMBL16487341 0.73 ALDH1A1 (0.50) XDHCYP1A2MAPTCYP3A4CYP2D6
SCHEMBL127566 0.72 HTR1B (0.52) NQO2MTNR1ATLR8SSTR2SSTR4
SCHEMBL15345359 0.72 TLR8 (0.49) MTNR1ATLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745586-B1 Aryl(alkyl) propylamides, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-03-08 EP disclosed
US-5760071-A AN UREA OR THIOUREA COMPOUNDS FOR TREATING MELATONINERGIC SYSTEM DISORDER, SLEEP DISORDER ADIR ET COMPAGNIE (FR) 1998-06-02 US disclosed
US-5731352-A THERAPY FOR DISORDERS OF THE MELATONINERGIC SYSTEM ADIR ET COMPAGNIE (FR) 1998-03-24 US disclosed
EP-0745586-A1 Aryl(alkyl) propylamides, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-12-04 EP disclosed