SCHEMBL8021973

SCHEMBL8021973

CCCCN(CCCN(CCCCCCCCN(CCCN(CCCC)C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 2/20 0.54
CA12 O43570 5/20 0.42
CA1 P00915 5/20 0.42
CA9 Q16790 4/20 0.42
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
MMP8 P22894 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CA2 P00918 2/20 0.37
CA7 P43166 1/20 0.37
HDAC3 O15379 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ZDHHC20 Q5W0Z9 2/20 0.35
ZDHHC2 Q9UIJ5 1/20 0.35
ALDH1A1 P00352 1/20 0.34
ALDH2 P05091 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14755630 0.96 CA14 (0.54) CA14CA12CA1CA9HDAC1
SCHEMBL1962811 0.94 CA14 (0.55) CA14CA12CA1CA9HDAC1
SCHEMBL136485 0.94 CA14 (0.55) CA14CA12CA1CA9HDAC1
SCHEMBL133198 0.94 CA14 (0.55) CA14CA12CA1CA9HDAC1
SCHEMBL140146 0.94 CA14 (0.55) CA14CA12CA1CA9HDAC1
SCHEMBL25969918 0.94 CA14 (0.54) CA14CA12CA1CA9HDAC1
SCHEMBL18163279 0.91 CA14 (0.53) CA14CA12CA1CA9HDAC1
SCHEMBL26616523 0.91 CA14 (0.53) CA14CA12CA1CA9HDAC1
SCHEMBL8285770 0.91 CA14 (0.51) CA14CA12CA1CA9HDAC1
SCHEMBL10226271 0.90 CA14 (0.49) CA14CA12CA1CA9HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114394-A Polyamine derivatives as radioprotective agents MERRELL PHARMACEUTICALS INC. (US) 2000-09-05 US disclosed
EP-0686142-B1 POLYAMINE DERIVATIVES AS RADIOPROTECTIVE AGENTS MERRELL PHARMA INC (US) 1998-12-30 EP disclosed
US-5753714-A ANTIPROTOZOA AGENTS MERRELL PHARMACEUTICALS INC. (US) 1998-05-19 US disclosed
EP-0686142-A1 POLYAMINE DERIVATIVES AS RADIOPROTECTIVE AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-12-13 EP disclosed
WO-1994019311-A1 POLYAMINE DERIVATIVES AS RADIOPROTECTIVE AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-09-01 WO disclosed
EP-0277635-B1 Novel polyamine derivatives MERRELL DOW PHARMA (US) 1994-01-05 EP disclosed
EP-0277635-A2 Novel polyamine derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-10 EP disclosed