SCHEMBL8022129

SCHEMBL8022129

CCOC(=O)C=CCC(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.59
MAPT P10636 4/20 0.53
ALDH1A1 P00352 4/20 0.47
CYP2D6 P10635 2/20 0.46
ALOX15 P16050 1/20 0.46
TTR P02766 1/20 0.42
DPP4 P27487 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CYP3A4 P08684 1/20 0.40
ATM Q13315 1/20 0.39
RAB9A P51151 1/20 0.38
MDM4 O15151 1/20 0.37
LMNA P02545 1/20 0.37
MDM2 Q00987 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25331608 0.83 HCAR2 (0.62) HCAR2MAPTALDH1A1CYP2D6ALOX15
SCHEMBL61548 0.83 HCAR2 (0.54) HCAR2MAPTALDH1A1TTRDPP4
SCHEMBL13990116 0.83 HCAR2 (0.54) HCAR2MAPTALDH1A1TTRDPP4
SCHEMBL4091546 0.83 HCAR2 (0.54) HCAR2MAPTALDH1A1TTRDPP4
SCHEMBL8925907 0.83 HCAR2 (0.54) HCAR2MAPTALDH1A1ALOX15TTR
SCHEMBL25331149 0.80 ATM (0.68) HCAR2MAPTALDH1A1CYP2D6ALOX15
SCHEMBL264771 0.79
SCHEMBL691584 0.79
SCHEMBL94678 0.79
SCHEMBL17019599 0.79 HCAR2 (0.67) HCAR2MAPTALDH1A1TTRDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4674894-A2 COPOLYMERS OF N-VINYLPYRROLIDONE WITH FUNCTIONALIZED MALEIC ACID MOIETIES Hemoteq AG (DE) 2026-01-07 EP disclosed
EP-4663688-A2 CROSSLINKERS Hemoteq AG (DE) 2025-12-17 EP disclosed
EP-4584243-B1 CROSSLINKERS HEMOTEQ AG (DE) 2025-11-05 EP disclosed
EP-4584243-A1 CROSSLINKERS Hemoteq AG (DE) 2025-07-16 EP disclosed
EP-4584245-A1 COPOLYMERS OF N-VINYLPYRROLIDONE WITH FUNCTIONALIZED MALEIC ACID MOIETIES Hemoteq AG (DE) 2025-07-16 EP disclosed
EP-4584244-A1 COPOLYMERS OF N-VINYLPYRROLIDONE WITH FUNCTIONALIZED MALEIC ACID MOIETIES Hemoteq AG (DE) 2025-07-16 EP disclosed
WO-2025056813-A1 COPOLYMERS OF N-VINYLPYRROLIDONE WITH FUNCTIONALIZED MALEIC ACID MOIETIES HEMOTEQ AG (DE) 2025-03-20 WO disclosed
WO-2025056815-A1 COPOLYMERS OF N-VINYLPYRROLIDONE WITH FUNCTIONALIZED MALEIC ACID MOIETIES HEMOTEQ AG (DE) 2025-03-20 WO disclosed
WO-2025056814-A1 CROSSLINKERS HEMOTEQ AG (DE) 2025-03-20 WO disclosed
EP-4524128-A1 BENZOPHENONE CROSSLINKERS Hemoteq AG (DE) 2025-03-19 EP disclosed
WO-2024070622-A1 CARBOXYL GROUP-CONTAINING ACRYLIC RUBBER COMPOSITION AND CROSSLINKED PRODUCT THEREOF 株式会社大阪ソーダ 2024-04-04 WO disclosed
EP-4223511-A1 CARBOXYL GROUP-CONTAINING ACRYLIC RUBBER COMPOSITION AND MULTILAYER BODY Osaka Soda Co., Ltd. (JP) 2023-08-09 EP disclosed
WO-2022071217-A1 CARBOXYL GROUP-CONTAINING ACRYLIC RUBBER COMPOSITION AND MULTILAYER BODY 株式会社大阪ソーダ 2022-04-07 WO disclosed
US-6106807-A Use of methylenemalondiester derivatives for the production of gas-containing microparticles for ultrasound diagnosis, as well as media that contain said particles SCHERING AKTIENGESELLSCHAFT (DE) 2000-08-22 US disclosed
EP-0804250-A1 USE OF METHYLENE MALONIC DIESTER DERIVATIVES IN THE PRODUCTION OF GAS-CONTAINING MICROPARTICLES FOR USE IN ULTRASOUND DIAGNOSTICS, AND AGENTS CONTAINING THESE PARTICLES SCHERING AKTIENGESELLSCHAFT (DE) 1997-11-05 EP disclosed
WO-1996025954-A1 USE OF METHYLENE MALONIC DIESTER DERIVATIVES IN THE PRODUCTION OF GAS-CONTAINING MICROPARTICLES FOR USE IN ULTRASOUND DIAGNOSTICS, AND AGENTS CONTAINING THESE PARTICLES SCHERING AKTIENGESELLSCHAFT (DE) 1996-08-29 WO disclosed