SCHEMBL8022200

SCHEMBL8022200

CN(C)C(=O)NC(=O)C#Cc1cccc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.51
GRM5 P41594 4/20 0.45
CYP1A2 P05177 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL667669 0.80 GFER (0.57) GFERGRM5
SCHEMBL8022201 0.76 GRM5 (0.44) GFERGRM5NPSR1
SCHEMBL14907878 0.74 GFER (0.51) GFERGRM5
SCHEMBL1751529 0.74 GFER (0.50) GFERGRM5
SCHEMBL2636049 0.73 GFER (0.55) GFERGRM5
SCHEMBL6563747 0.72 CA12 (0.51) GFERGRM5
SCHEMBL14907954 0.71 GFER (0.51) GFERCYP1A2
SCHEMBL29941936 0.71 GFER (0.47) GFERGRM5
SCHEMBL28909500 0.71 GFER (0.47) GFERGRM5
SCHEMBL26343014 0.70 GFER (0.46) GFERGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6069247-A REACTING AN ACETYLENECARBOXY AMIDE AND AN ARYL OR HETEROCYCLYL HALIDE OR A GROUP ENHANCING THE ELECTROPHILICITY OF THE ATOM TO WHICH IT IS ATTACHED FOR DISPLACEMENT; USING A PALLADIUM COMPOUND CATALYST, A BASE AND AN ACID ELI LILLY AND COMPANY (US) 2000-05-30 US disclosed