SCHEMBL8022210

SCHEMBL8022210

Cc1cccc(-c2nc3ccccc3n2Cc2ccccc2I)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.68
MAPT P10636 7/20 0.63
GAA P10253 1/20 0.55
ALDH1A1 P00352 3/20 0.51
PDE6D O43924 1/20 0.51
ALDH2 P05091 1/20 0.51
ALDH3A1 P30838 1/20 0.51
KMT2A Q03164 4/20 0.50
MEN1 O00255 3/20 0.50
LMNA P02545 4/20 0.48
TSHR P16473 3/20 0.48
HSD17B10 Q99714 2/20 0.48
NPC1 O15118 1/20 0.47
GALR3 O60755 1/20 0.47
NR2F2 P24468 1/20 0.47
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 5/20 0.46
NPSR1 Q6W5P4 4/20 0.46
HTT P42858 3/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8023982 0.85 TP53 (0.68) TP53MAPTGAAALDH1A1PDE6D
SCHEMBL8022017 0.85 TP53 (0.72) TP53MAPTGAAALDH1A1PDE6D
SCHEMBL29412044 0.81 TP53 (1.00) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL8010677 0.80 KDM4E (0.56) TP53MAPTGAAALDH1A1KMT2A
SCHEMBL8025719 0.79 TP53 (0.67) TP53MAPTGAAALDH1A1PDE6D
SCHEMBL8022045 0.78 TP53 (0.82) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL8022230 0.78 TP53 (0.74) TP53MAPTGAAALDH1A1PDE6D
SCHEMBL8027160 0.76 TP53 (0.83) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL8021682 0.75 TP53 (0.77) TP53MAPTGAAALDH1A1PDE6D
Bromide SCHEMBL8021395 0.75 TP53 (0.77) TP53MAPTGAAALDH1A1PDE6D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6030992-A ANTAGONISTS FOR THE BINDING OF NEUROKININ-2 RECEPTOR; SLEEP DISORDERS; BENZIMIDES, 2- OR 3-ALKOXYBENZIMIDES AND 2,3-DIALKOXYBENZIMIDES ELI LILLY AND COMPANY (US) 2000-02-29 US disclosed
US-6025379-A A SUBSTITUTED BENZIMIDAZOLE, TACHYKININ RECEPTOR ANTAGONISTS, ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed
WO-1997033873-A1 METHODS OF TREATING OR PREVENTING INTERSTITIAL CYSTITIS ELI LILLY AND COMPANY (US) 1997-09-18 WO disclosed
WO-1997031635-A1 METHODS OF TREATING OR PREVENTING SLEEP APNEA ELI LILLY AND COMPANY (US) 1997-09-04 WO disclosed
US-5552426-A NERVOUS SYSTEM DISORDERS USING IMIDAZOLE DERIVITIVES ELI LILLY AND COMPANY (US) 1996-09-03 US disclosed
EP-0694535-A1 Non-peptidyl tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-01-31 EP disclosed