SCHEMBL8022502

SCHEMBL8022502

O=C(c1cccc2ccccc12)N1CC(CC(O)c2ccccc2)C(CN2CCC(c3ccc(F)cc3)CC2)C1

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.65
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651239 0.88 CCR5 (0.65) CCR5KDM4EALDH1A1TP53TSHR
SCHEMBL7658040 0.88 CCR5 (0.65) CCR5KDM4EALDH1A1TP53TSHR
SCHEMBL7650129 0.87 CCR5 (0.69) CCR5KDM4EALDH1A1TP53TSHR
SCHEMBL7650468 0.86 CCR5 (0.64) CCR5KDM4EALDH1A1TP53TSHR
SCHEMBL7650472 0.85 CCR5 (0.67) CCR5KDM4EALDH1A1TP53TSHR
SCHEMBL7833271 0.85 CCR5 (0.89) CCR5
SCHEMBL7652090 0.85 CCR5 (0.70) CCR5KDM4EALDH1A1TP53TSHR
SCHEMBL7655471 0.85 CCR5 (0.67) CCR5KDM4EALDH1A1
SCHEMBL8024899 0.84 CCR5 (0.66) CCR5KDM4EALDH1A1TP53TSHR
SCHEMBL7687323 0.84 CCR5 (0.64) CCR5KDM4EALDH1A1TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000051609-A1 3-ALKYL SUBSTITUTED PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-09-08 WO disclosed