SCHEMBL8024907

SCHEMBL8024907

CC1(C)CSc2ccccc2N(c2ccccc2)C1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
ELANE P08246 3/20 0.41
SLC6A2 P23975 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HPGD P15428 1/20 0.39
PGR P06401 1/20 0.39
CACNA1B Q00975 1/20 0.37
APBA1 Q02410 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
THPO P40225 1/20 0.37
CES2 O00748 1/20 0.37
BCHE P06276 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024775 0.82 SLC6A2 (0.49) ALDH1A1ELANESLC6A2NPSR1MEN1
SCHEMBL8014427 0.76 SLC6A2 (0.52) ALDH1A1ELANESLC6A2MEN1KMT2A
SCHEMBL8027951 0.76 NOTUM (0.30)
SCHEMBL10353018 0.71 GSK3B (0.55) ALDH1A1NPSR1MEN1KMT2ASMN1; SMN2
SCHEMBL11421115 0.71 ALDH1A1 (0.46) ALDH1A1ELANESLC6A2MEN1KMT2A
SCHEMBL8013849 0.70 TMEM97 (0.40) ALDH1A1SLC6A2MEN1KMT2ASMN1; SMN2
SCHEMBL8014417 0.70 ALDH1A1 (0.44) ALDH1A1ELANESLC6A2NPSR1MEN1
SCHEMBL10855612 0.69 ALDH1A1 (0.51) ALDH1A1ELANEMEN1KMT2ASMN1; SMN2
SCHEMBL12997888 0.68 PGR (0.65) ALDH1A1ELANEMEN1KMT2APGR
SCHEMBL7372104 0.68 PGR (0.65) ALDH1A1ELANEMEN1KMT2APGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792268-B1 HYPOLIPIDEMIC BENZOTHIAZEPINES WELLCOME FOUND (GB) 2000-02-23 EP claimed
US-5998400-A Hypolipidemic benzothiazepines GLAXO WELLCOME INC. (US) 1999-12-07 US claimed
EP-0792268-A1 HYPOLIPIDEMIC BENZOTHIAZEPINES THE WELLCOME FOUNDATION LIMITED (GB) 1997-09-03 EP claimed
WO-1996016051-A1 HYPOLIPIDEMIC BENZOTHIAZEPINES THE WELLCOME FOUNDATION LIMITED (GB) 1996-05-30 WO claimed
EP-0792268-B1 HYPOLIPIDEMIC BENZOTHIAZEPINES WELLCOME FOUND (GB) 2000-02-23 EP disclosed
EP-0971744-A2 COMBINATION THERAPY EMPLOYING ILEAL BILE ACID TRANSPORT INHIBITING BENZOTHIEPINES AND HMG Co-A REDUCTASE INHIBITORS G.D. SEARLE & CO. (US) 2000-01-19 EP disclosed
US-5998400-A Hypolipidemic benzothiazepines GLAXO WELLCOME INC. (US) 1999-12-07 US disclosed
WO-1998040375-A2 COMBINATION OF ILEAL BILE ACID TRANSPORT INHIBITING BENZOTHIEPINES AND HMG Co-A REDUCTASE INHIBITORS G.D. SEARLE & CO. (US) 1998-09-17 WO disclosed
EP-0792268-A1 HYPOLIPIDEMIC BENZOTHIAZEPINES THE WELLCOME FOUNDATION LIMITED (GB) 1997-09-03 EP disclosed
WO-1996016051-A1 HYPOLIPIDEMIC BENZOTHIAZEPINES THE WELLCOME FOUNDATION LIMITED (GB) 1996-05-30 WO disclosed