SCHEMBL8026608

SCHEMBL8026608

O=C1CCCC=C1c1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.46
BRD4 O60885 1/20 0.45
KDM4E B2RXH2 3/20 0.42
GAA P10253 2/20 0.42
ALPL P05186 1/20 0.42
CYP2A6 P11509 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
GALR1 P47211 1/20 0.38
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
LMNA P02545 2/20 0.38
HTT P42858 2/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PARP1 P09874 1/20 0.36
HPGD P15428 3/20 0.36
HSD17B10 Q99714 2/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28422058 0.79 CYP2A6 (0.40) CYP2A6MAOAMAOBMAPTNPSR1
SCHEMBL28777035 0.75 GRM2 (0.46) PTPN1BRD4KDM4EGAAALPL
SCHEMBL6823018 0.71 PTPN1 (0.49) PTPN1KDM4EGAAMAOBALDH1A1
SCHEMBL11502520 0.71 MAPT (0.41) CYP2A6MAOAMAOBALDH1A1MAPT
SCHEMBL1943625 0.71 BACE1 (0.39) PTPN1BRD4KDM4ECYP2A6MAOA
SCHEMBL3160653 0.70 TDP1 (0.46) BRD4KDM4EGALR1ALDH1A1HPGD
SCHEMBL8027778 0.70 GSTP1 (0.46) MAOBNISCH
SCHEMBL4276998 0.70 PTPN1 (0.43) PTPN1BRD4KDM4EGAAALPL
SCHEMBL9620885 0.69 ELANE (0.46) KDM4EGALR1ALDH1A1HPGDMEN1
SCHEMBL30527944 0.69 PTPN1 (0.49) PTPN1KDM4EGAAALPLMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3746436-A1 FUSED RING COMPOUNDS F. Hoffmann-La Roche AG (CH) 2020-12-09 EP disclosed
WO-2020035031-A1 FUSED RING COMPOUNDS GENENTECH, INC. (US) 2020-02-20 WO disclosed
WO-2000064908-A1 N-TRI OR DI-ALKYLSILYL( PERFLUOROAL KANESULPHONYL) IMIDE DERIVATIVES, PREPARATION AND USE RHODIA CHIMIE (FR) 2000-11-02 WO disclosed