SCHEMBL8027345

SCHEMBL8027345

Cc1sc(C)c2c1CCc1cnn(C)c1-2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 17/20 1.00
DRD2 P14416 11/20 1.00
CCNC P24863 2/20 0.49
CDK8 P49336 2/20 0.49
CDK19 Q9BWU1 2/20 0.49
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8022012 0.98 DRD4 (0.97) DRD4DRD2CCNCCDK8CDK19
SCHEMBL8022043 0.91 DRD4 (1.00) DRD4DRD2CCNCCDK8CDK19
Hydrochloric Acid SCHEMBL8011148 0.89 DRD4 (0.97) DRD4DRD2CCNCCDK8CDK19
SCHEMBL7246869 0.82 DRD4 (0.68) DRD4DRD2CCNCCDK8CDK19
SCHEMBL7241539 0.81 CCNC (0.72) DRD4DRD2CCNCCDK8CDK19
SCHEMBL7241940 0.77 DRD2 (0.61) DRD4DRD2CCNCCDK8CDK19
SCHEMBL9212631 0.71 DRD4 (0.55) DRD4DRD2CCNCCDK8CDK19
SCHEMBL7248682 0.69 DRD4 (0.52) DRD4DRD2CCNCCDK8CDK19
SCHEMBL9222650 0.69 DRD2 (0.53) DRD4DRD2CCNCCDK8CDK19
SCHEMBL7246960 0.69 CCNC (0.52) DRD4DRD2CCNCCDK8CDK19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6034252-A Substituted thienocycloalkylpyrazoles: dopamine receptor subtype specific ligands NEUROGEN CORPORATION (US) 2000-03-07 US claimed