SCHEMBL9212631

SCHEMBL9212631

Cc1n[nH]c2c1-c1c(cnn1C)CC2

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 10/20 0.55
DRD2 P14416 9/20 0.55
CCNC P24863 2/20 0.40
CDK8 P49336 2/20 0.40
CDK19 Q9BWU1 2/20 0.40
FLT3 P36888 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9222650 0.72 DRD2 (0.53) DRD4DRD2CCNCCDK8CDK19
SCHEMBL8027345 0.71 DRD4 (1.00) DRD4DRD2CCNCCDK8CDK19
SCHEMBL9221790 0.70 CCNA2 (0.47) DRD4DRD2
SCHEMBL9219954 0.70 DRD4 (0.55) DRD4DRD2CCNCCDK8CDK19
Hydrochloric Acid SCHEMBL8022012 0.70 DRD4 (0.97) DRD4DRD2CCNCCDK8CDK19
SCHEMBL21614788 0.66 DRD2 (0.49) DRD4DRD2CCNCCDK8CDK19
SCHEMBL8022043 0.66 DRD4 (1.00) DRD4DRD2CCNCCDK8CDK19
Hydrochloric Acid SCHEMBL8011148 0.65 DRD4 (0.97) DRD4DRD2CCNCCDK8CDK19
SCHEMBL7246869 0.64 DRD4 (0.68) DRD4DRD2CCNCCDK8CDK19
SCHEMBL13085158 0.64 DRD2 (0.50) DRD4DRD2CCNCCDK8CDK19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276833-B1 Dipyrazoles useful as bronchodilators MERRELL DOW PHARMA (US) 1995-02-15 EP disclosed
EP-0276833-A2 Dipyrazoles useful as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP disclosed
US-4734430-A Dipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed