SCHEMBL8028243

SCHEMBL8028243

O=S(=O)(c1cccc(Cl)c1)c1nnn2c1ncc1ccsc12

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 18/20 0.59
RXFP1 Q9HBX9 5/20 0.55
MAPT P10636 3/20 0.55
GAA P10253 1/20 0.54
POLB P06746 1/20 0.51
TP53 P04637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026985 0.87 HTR6 (0.46) HTR6RXFP1MAPTGAA
SCHEMBL8018264 0.86 HTR6 (0.52) HTR6RXFP1MAPTTP53
SCHEMBL8019100 0.81 HTR6 (0.57) HTR6RXFP1MAPTGAATP53
SCHEMBL8019082 0.80 HTR6 (0.48) HTR6RXFP1MAPTPOLBTP53
SCHEMBL8028875 0.79 HTR6 (0.61) HTR6RXFP1MAPTGAAPOLB
SCHEMBL8021774 0.79 RXFP1 (0.64) HTR6RXFP1MAPTGAATP53
SCHEMBL8019579 0.73 HTR6 (0.76) HTR6RXFP1MAPTTP53
SCHEMBL8019326 0.71 HTR6 (0.98) HTR6RXFP1MAPTGAAPOLB
SCHEMBL8027278 0.70 HTR6 (0.85) HTR6RXFP1MAPTGAAPOLB
SCHEMBL8030163 0.69 HTR6 (1.00) HTR6RXFP1MAPTGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed