SCHEMBL8028353

SCHEMBL8028353

COc1cc(C#N)c(C(=O)N(C)C(=O)NC2CC2)c([N+](=O)O)c1O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
ACHE P22303 4/20 0.37
ALDH1A1 P00352 5/20 0.34
MAPT P10636 5/20 0.34
KDM4E B2RXH2 4/20 0.34
GAA P10253 2/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
TAS1R2 Q8TE23 1/20 0.34
DRD2 P14416 1/20 0.34
MELK Q14680 1/20 0.34
ERN1 O75460 1/20 0.32
POLB P06746 2/20 0.32
LMNA P02545 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028359 0.73 SMN1; SMN2 (0.35) ALDH1A1MAPTKDM4EGAATAS1R3
SCHEMBL8035126 0.68 ALDH1A1 (0.40) ALDH1A1MAPTKDM4EGAAERN1
SCHEMBL12082469 0.67 COMT (0.42) ALDH1A1MAPTKDM4EPOLBLMNA
SCHEMBL12082492 0.67 SMN1; SMN2 (0.46) ALDH1A1MAPTKDM4EGAAERN1
SCHEMBL12082409 0.66 EGFR (0.37) ALDH1A1MAPTKDM4EERN1POLB
SCHEMBL12082329 0.65 EGFR (0.37) ALDH1A1MAPTKDM4EERN1POLB
SCHEMBL12082493 0.65 EGFR (0.37) ALDH1A1MAPTKDM4EERN1POLB
SCHEMBL12082487 0.65 EGFR (0.42) ALDH1A1MAPTKDM4EGAAERN1
SCHEMBL12082451 0.65 MAPT (0.40) ALDH1A1MAPTKDM4EGAAERN1
SCHEMBL8031695 0.64 ALDH1A1 (0.43) ALDH1A1MAPTKDM4EGAATAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed