SCHEMBL8028362

SCHEMBL8028362

CN(C(=O)c1ccc2c(c1)nc(Cc1ccc(C#N)cc1)n2C)c1cccnc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 7/20 0.50
F2 P00734 4/20 0.47
TRPV1 Q8NER1 1/20 0.45
TXK P42681 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
CNR2 P34972 3/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
ACSL1 P33121 1/20 0.40
PDK1 Q15118 1/20 0.40
AURKA O14965 1/20 0.40
MAP4K4 O95819 1/20 0.40
CHEK2 O96017 1/20 0.40
PRKCG P05129 1/20 0.40
PHKG2 P15735 1/20 0.40
MARK3 P27448 1/20 0.40
FLT3 P36888 1/20 0.40
CSNK1A1 P48729 1/20 0.40
CSNK1D P48730 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7247078 0.92 F2 (0.51) ITKF2TRPV1TXKHDAC1
SCHEMBL8028940 0.90 ITK (0.60) ITKF2TXKACSL1PDK1
Hydrochloric Acid SCHEMBL8026382 0.86 F2 (0.62) F2
SCHEMBL8026572 0.84 ITK (0.57) ITKF2TXKCNR2ACSL1
SCHEMBL8016085 0.83 F2 (0.47) ITKF2TXKHDAC6CNR2
SCHEMBL8016095 0.81 F2 (0.48) ITKF2TXKHDAC1HDAC6
SCHEMBL8026270 0.81 F2 (0.51) ITKF2HDAC1HDAC6CNR2
SCHEMBL8028885 0.80 HDAC6 (0.46) F2HDAC1HDAC6CNR2BCHE
SCHEMBL7246372 0.79 PDK1 (0.51) ITKF2HDAC1HDAC6PDK1
Hydrochloric Acid SCHEMBL7247385 0.78 F2 (0.66) F2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060166-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS Boehringer Ingelheim Pharma KG (DE) 2000-12-20 EP disclosed
US-6114532-A ANTICOAGULANT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-05 US disclosed
WO-1999040072-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-08-12 WO disclosed