SCHEMBL8028787

SCHEMBL8028787

CN(C(=O)N1CCc2ccccc21)c1ccc2c(c1)nc(Cc1ccc(C#N)cc1)n2C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.42
USP2 O75604 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HSD17B10 Q99714 2/20 0.42
ALOX15 P16050 1/20 0.42
MAPK1 P28482 1/20 0.42
ITK Q08881 7/20 0.41
AURKA O14965 1/20 0.41
MAP4K4 O95819 1/20 0.41
CHEK2 O96017 1/20 0.41
PRKCG P05129 1/20 0.41
PHKG2 P15735 1/20 0.41
MARK3 P27448 1/20 0.41
FLT3 P36888 1/20 0.41
CSNK1A1 P48729 1/20 0.41
CSNK1D P48730 1/20 0.41
CLK2 P49760 1/20 0.41
GSK3B P49841 1/20 0.41
IRAK1 P51617 1/20 0.41
RPS6KA3 P51812 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8032368 0.85 F2 (0.58) F2USP2ALDH1A1HSD17B10ALOX15
SCHEMBL8028430 0.82 CNR2 (0.57) F2ITKAURKAMAP4K4CHEK2
SCHEMBL8026604 0.78 F2 (0.47) F2ALDH1A1HSD17B10ITKAURKA
SCHEMBL8031763 0.76 PKM (0.52) USP2ALDH1A1HSD17B10ALOX15MAPK1
SCHEMBL8026572 0.76 ITK (0.57) F2ITKAURKAMAP4K4CHEK2
SCHEMBL8028940 0.75 ITK (0.60) F2ITKAURKAMAP4K4CHEK2
SCHEMBL8016797 0.73 F2 (0.71) F2CNR2ACSL1POLBMEN1
SCHEMBL8139393 0.73 CNR2 (0.59) USP2ITKCNR2CNR1POLB
SCHEMBL7115133 0.71 ITK (0.47) F2ITKAURKAMAP4K4CHEK2
SCHEMBL8032935 0.70 F2 (0.49) F2USP2ITKACSL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114532-A ANTICOAGULANT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-05 US disclosed