SCHEMBL8026604

SCHEMBL8026604

CN(C(=O)NCc1ccccc1)c1ccc2c(c1)nc(Cc1ccc(C#N)cc1)n2C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 2/20 0.47
HDAC1 Q13547 5/20 0.46
HDAC6 Q9UBN7 2/20 0.46
ITK Q08881 8/20 0.45
TXK P42681 1/20 0.45
ACSL1 P33121 1/20 0.45
AURKA O14965 1/20 0.44
MAP4K4 O95819 1/20 0.44
CHEK2 O96017 1/20 0.44
PRKCG P05129 1/20 0.44
PHKG2 P15735 1/20 0.44
MARK3 P27448 1/20 0.44
FLT3 P36888 1/20 0.44
CSNK1A1 P48729 1/20 0.44
CSNK1D P48730 1/20 0.44
CLK2 P49760 1/20 0.44
GSK3B P49841 1/20 0.44
IRAK1 P51617 1/20 0.44
RPS6KA3 P51812 1/20 0.44
NEK4 P51957 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8015782 0.84 RORC (0.58) HDAC1HDAC6RORC
SCHEMBL8028940 0.80 ITK (0.60) F2ITKTXKACSL1AURKA
SCHEMBL8026572 0.80 ITK (0.57) F2ITKTXKACSL1AURKA
SCHEMBL8028430 0.79 CNR2 (0.57) F2ITKACSL1AURKAMAP4K4
SCHEMBL6637343 0.79 HDAC6 (0.49) F2HDAC1HDAC6ITKTXK
SCHEMBL8016797 0.79 F2 (0.71) F2ACSL1CNR2TSHR
SCHEMBL7120171 0.78 HDAC1 (0.43) F2HDAC1HDAC6ITKTXK
SCHEMBL8032935 0.78 F2 (0.49) F2HDAC1HDAC6ITKACSL1
SCHEMBL8028787 0.78 F2 (0.42) F2ITKTXKACSL1AURKA
SCHEMBL8028885 0.78 HDAC6 (0.46) F2HDAC1HDAC6ACSL1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114532-A ANTICOAGULANT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-05 US disclosed