SCHEMBL8028817

SCHEMBL8028817

Cc1noc(-c2noc(N)n2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.48
LMNA P02545 1/20 0.44
THRB P10828 1/20 0.44
RECQL P46063 1/20 0.42
NOTUM Q6P988 1/20 0.42
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
BCHE P06276 1/20 0.34
NPC1 O15118 5/20 0.33
RAB9A P51151 5/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
ACE2 Q9BYF1 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
HDAC3 O15379 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL558663 0.79
SCHEMBL6003977 0.74 RECQL (0.58) RECQLNOTUMACE2
SCHEMBL981283 0.65 ACHE (1.00) ACHELMNATHRBTP53MAPT
SCHEMBL29164847 0.64 ACHE (0.42) ACHELMNATP53MAPTBCHE
SCHEMBL30822733 0.64 ACHE (0.42) ACHELMNATP53MAPTBCHE
SCHEMBL16597159 0.64 ACHE (0.50) ACHEBCHE
SCHEMBL2618901 0.64 LMNA (0.66) ACHELMNATHRBTP53MAPT
SCHEMBL21547867 0.64 PPARA (0.49) ACHELMNATHRBTP53NPC1
SCHEMBL13415305 0.64 ACHE (0.80) ACHELMNATHRBTP53MAPT
SCHEMBL2618848 0.63 LMNA (0.69) ACHELMNATHRBTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663171-A FOR USE IN HUMANS OR ANIMALS MERCK & CO., INC. (US) 1997-09-02 US claimed
US-6121325-A Naphthyl compounds promote release of growth hormone MERCK & CO., INC. (US) 2000-09-19 US disclosed
US-5663171-A FOR USE IN HUMANS OR ANIMALS MERCK & CO., INC. (US) 1997-09-02 US disclosed