SCHEMBL8028826

SCHEMBL8028826

CC(=O)Oc1ccc(C=CC(=O)OCC(OC(=O)C=Cc2ccc(OC(C)=O)c(OC(C)=O)c2)C(=O)O)cc1OC(C)=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 9/20 0.58
KDM4E B2RXH2 5/20 0.55
MAPT P10636 5/20 0.55
RECQL P46063 3/20 0.55
HTT P42858 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
GLA P06280 1/20 0.55
GAA P10253 3/20 0.53
JAK2 O60674 1/20 0.53
ALDH1A1 P00352 1/20 0.53
JUN P05412 2/20 0.50
NFKB1 P19838 1/20 0.50
MMP1 P03956 4/20 0.48
AKR1C3 P42330 1/20 0.47
AKR1C2 P52895 1/20 0.47
TDP1 Q9NUW8 3/20 0.46
POLB P06746 2/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
CYP1A2 P05177 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8031841 0.90 KDM4E (0.60) ALOX5KDM4EMAPTRECQLHTT
SCHEMBL30075809 0.83 TP53 (0.60) ALOX5KDM4EMAPTRECQLHTT
SCHEMBL8028622 0.82 ALOX5 (0.56) ALOX5KDM4EMAPTRECQLHTT
SCHEMBL8034404 0.81 ALOX5 (0.79) ALOX5KDM4EMAPTHTTSMN1; SMN2
SCHEMBL8019019 0.80 ALOX5 (0.54) ALOX5KDM4EMAPTRECQLHTT
SCHEMBL8030403 0.80 ALOX5 (0.54) ALOX5KDM4EMAPTRECQLHTT
SCHEMBL8019021 0.80 ALOX5 (0.54) ALOX5KDM4EMAPTRECQLHTT
SCHEMBL8019035 0.79 TDP1 (0.71) ALOX5KDM4EMAPTRECQLSMN1; SMN2
SCHEMBL25804735 0.79 TDP1 (0.71) ALOX5KDM4EMAPTRECQLSMN1; SMN2
SCHEMBL8028624 0.77 KDM4E (0.60) ALOX5KDM4EMAPTRECQLHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000063152-A1 ACETYLATED AND RELATED ANALOGUES OF CHICORIC ACID AS HIV INTEGRASE INHIBITORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-10-26 WO disclosed