Dioxane

Dioxane

SCHEMBL8029153

C1COCCO1.O=C(O)Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.53
SRD5A2 P31213 2/20 0.50
BCL9 O00512 1/20 0.50
CTNNB1 P35222 1/20 0.50
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
PKM P14618 1/20 0.49
MEN1 O00255 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
PAX8 Q06710 1/20 0.46
RAB9A P51151 1/20 0.46
POLB P06746 1/20 0.46
KCNJ1 P48048 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
AKR1C3 P42330 1/20 0.46
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tetrahydrofuran SCHEMBL3720210 0.94 BCL9 (0.51) GAASRD5A2BCL9CTNNB1KMT2A
Tetrahydrofuran SCHEMBL1273145 0.94 BCL9 (0.51) GAASRD5A2BCL9CTNNB1KMT2A
SCHEMBL27544786 0.92 BCL9 (0.50) GAASRD5A2BCL9CTNNB1KMT2A
SCHEMBL26375 0.89 GAA (0.62) GAASRD5A2BCL9CTNNB1KMT2A
Cyclohexane SCHEMBL30739999 0.88 GAA (0.57) GAASRD5A2BCL9CTNNB1KMT2A
Bromide SCHEMBL30468845 0.88 GAA (0.61) GAASRD5A2BCL9CTNNB1KMT2A
Bicarbonate SCHEMBL7985678 0.88 GAA (0.61) GAASRD5A2BCL9CTNNB1KMT2A
Hydrochloric Acid SCHEMBL7895039 0.88 GAA (0.61) GAASRD5A2BCL9CTNNB1KMT2A
Bicarbonate SCHEMBL9330234 0.84 GAA (0.57) GAASRD5A2BCL9CTNNB1KMT2A
SCHEMBL26654348 0.84 GAA (0.57) GAASRD5A2BCL9CTNNB1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127372-A FOR TREATMENT OR PREVENTION OF VIRAL DISEASES, ESPECIALLY AIDS OR HIV VERTEX PHARMACEUTICALS, INCORPORATED (US) 2000-10-03 US disclosed
EP-0749421-B1 SULPHONAMIDE DERIVATIVES AS ASPARTYL PROTEASE INHIBITORS VERTEX PHARMA (US) 1999-09-15 EP disclosed
EP-0749421-A1 SULPHONAMIDE DERIVATIVES AS ASPARTYL PROTEASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 1996-12-27 EP disclosed
WO-1995024385-A1 SULPHONAMIDE DERIVATIVES AS ASPARTYL PROTEASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-09-14 WO disclosed