SCHEMBL8029322

SCHEMBL8029322

CCCCCOC1C(=O)c2cc(OCc3ccc4ccccc4n3)cnc2CC1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.53
CYSLTR1 Q9Y271 10/20 0.50
CYSLTR2 Q9NS75 7/20 0.50
MAPK1 P28482 2/20 0.44
ALOX5 P09917 2/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
CYP2C19 P33261 1/20 0.44
HIF1A Q16665 1/20 0.44
MEN1 O00255 1/20 0.44
GMNN O75496 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029325 1.00 GPBAR1 (0.53) GPBAR1CYSLTR1CYSLTR2MAPK1ALOX5
SCHEMBL8029321 1.00 GPBAR1 (0.53) GPBAR1CYSLTR1CYSLTR2MAPK1ALOX5
SCHEMBL8032680 0.85 GPBAR1 (0.49) GPBAR1CYSLTR1CYSLTR2MAPK1ALOX5
SCHEMBL8029124 0.85 GPBAR1 (0.49) GPBAR1CYSLTR1CYSLTR2MAPK1ALOX5
SCHEMBL8032678 0.85 GPBAR1 (0.49) GPBAR1CYSLTR1CYSLTR2MAPK1ALOX5
SCHEMBL8461158 0.85 CYSLTR1 (0.49) GPBAR1CYSLTR1CYSLTR2ALOX5
SCHEMBL8461147 0.85 CYSLTR1 (0.49) GPBAR1CYSLTR1CYSLTR2ALOX5
SCHEMBL8461154 0.85 CYSLTR1 (0.49) GPBAR1CYSLTR1CYSLTR2ALOX5
SCHEMBL8032722 0.77 CYSLTR1 (0.49) GPBAR1CYSLTR1CYSLTR2ALOX5ALOX5AP
SCHEMBL8462463 0.76 LTB4R (0.49) GPBAR1CYSLTR1CYSLTR2ALOX5ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166031-A Substituted tetralins, chromans and related compounds in the treatment of asthma PFIZER INC, (US) 2000-12-26 US disclosed
WO-1989003681-A1 SUBSTITUTED TETRALINS, CHROMANS AND RELATED COMPOUNDS IN THE TREATMENT OF ASTHMA PFIZER INC. (US) 1989-05-05 WO disclosed