SCHEMBL8029620

SCHEMBL8029620

CC(C)Oc1ccc(CN2CCN(CC3CCc4ccccc4O3)CC2)cc1

nearest known ligand 0.71

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.71
HTR1A P08908 5/20 0.71
ADRA2A P08913 1/20 0.71
ADRA2B P18089 1/20 0.71
ADRA2C P18825 1/20 0.71
FAAH O00519 1/20 0.45
ABCB1 P08183 1/20 0.43
HRH3 Q9Y5N1 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029651 0.88 SIGMAR1 (0.76) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8029628 0.84 SIGMAR1 (0.81) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL31061719 0.84 SIGMAR1 (1.00) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8031431 0.84 SIGMAR1 (1.00) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8029887 0.83 SIGMAR1 (0.83) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8035775 0.82 SIGMAR1 (0.81) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8031447 0.82 SIGMAR1 (0.81) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8033233 0.79 SIGMAR1 (0.76) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8031492 0.79 SIGMAR1 (0.76) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8029650 0.79 SIGMAR1 (0.71) SIGMAR1HTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0702010-B1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-03-15 EP disclosed
US-5668138-A AFFINITY FOR SIGMA RECEPTORS, CENTRAL NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-09-16 US disclosed
EP-0702010-A1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-03-20 EP disclosed