SCHEMBL8029685

SCHEMBL8029685

N#Cc1ccc(N)c(CN2CC[C@@H](C(N)=O)C2=O)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 3/20 0.35
SIRT1 Q96EB6 3/20 0.35
F10 P00742 7/20 0.35
F2 P00734 6/20 0.35
PROC P04070 2/20 0.34
PRSS1 P07477 2/20 0.34
PLG P00747 1/20 0.34
KDM2B Q8NHM5 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
ALDH1A1 P00352 3/20 0.33
DPP4 P27487 2/20 0.33
KDM4E B2RXH2 2/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PGGT1B P53609 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417913 1.00 SIRT2 (0.35) SIRT2SIRT1F10F2PROC
SCHEMBL8029146 0.88 SIRT2 (0.35) SIRT2SIRT1F10F2PROC
SCHEMBL8042725 0.88 SIRT2 (0.35) SIRT2SIRT1F10F2PROC
SCHEMBL8039167 0.87 HCRTR1 (0.39) SIRT2SIRT1F10F2DPP4
SCHEMBL7423151 0.84 KDM4E (0.35) F10F2PROCPRSS1PLG
SCHEMBL7424077 0.84 KDM4E (0.35) F10F2PROCPRSS1PLG
Hydrochloric Acid SCHEMBL8040100 0.83 KDM4E (0.35) F10F2PROCPRSS1PLG
Hydrochloric Acid SCHEMBL7423721 0.83 KDM4E (0.35) F10F2PROCPRSS1PLG
SCHEMBL27461354 0.82 KDM4E (0.34) F10F2PROCPRSS1PLG
SCHEMBL7424934 0.82 FNTA (0.44) DPP4FNTAFNTBPGGT1BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6034093-A Substituted sulfonic acid N-[(aminoiminomethyl)phenylalkyl]-azaheterocyclylamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 2000-03-07 US disclosed