SCHEMBL8030987

SCHEMBL8030987

N=C(N)c1ccc(N2CCCC2=O)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.68
HPGD P15428 6/20 0.59
F2 P00734 3/20 0.57
PRSS1 P07477 3/20 0.57
F10 P00742 2/20 0.57
PRSS2 P07478 2/20 0.53
PRSS3 P35030 2/20 0.53
TMPRSS6 Q8IU80 2/20 0.53
ST14 Q9Y5Y6 2/20 0.53
GRIN2D O15399 1/20 0.53
GRIN3B O60391 1/20 0.53
GRIN1 Q05586 1/20 0.53
GRIN2A Q12879 1/20 0.53
GRIN2B Q13224 1/20 0.53
GRIN2C Q14957 1/20 0.53
GRIN3A Q8TCU5 1/20 0.53
NPC1 O15118 6/20 0.52
RAB9A P51151 5/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
TSHR P16473 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4418893 0.85 ALDH1A1 (0.75) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL11142367 0.82 ALDH1A1 (0.74) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL70639 0.81 ALDH1A1 (1.00) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL6236939 0.80 ALDH1A1 (0.68) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL78465 0.78 ALDH1A1 (0.65) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL322211 0.78 ALDH1A1 (0.93) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL457785 0.78 ALDH1A1 (0.75) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL12359037 0.78 ALDH1A1 (0.75) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL27350108 0.78 F2 (0.55) ALDH1A1F2PRSS1F10PRSS2
SCHEMBL1656668 0.77 ALDH1A1 (0.68) ALDH1A1HPGDNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691953-B1 1-AMIDINOPHENYL-PYRROLIDONES/ PIPERIDINONES AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2000-08-02 EP disclosed
US-6037365-A ANTIINFLAMMATORY AND ANTIMETASTASIS AGENTS; CARDIOVASCULAR DISORDERS, ARTERIOSCLEROSIS G.D. SEARLE & CO. (US) 2000-03-14 US disclosed
US-5872122-A Pyrimidinylamidino β-amino acid derivatives useful as inhibitors of platelet aggregation MONSANTO COMPANY (US) 1999-02-16 US disclosed
US-5721366-A PHENYLAMIDINE DERIVATIVES G. D. SEARLE & CO (US) 1998-02-24 US disclosed