SCHEMBL8032018

SCHEMBL8032018

O=C(O)C(O)C(O)C(=O)ON1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
NFKB1 P19838 1/20 0.36
CYP2C19 P33261 1/20 0.36
DPP7 Q9UHL4 1/20 0.32
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5874105 0.92 ALDH1A1 (0.33)
SCHEMBL2786080 0.89 HTT (0.30)
SCHEMBL27576738 0.89 HTT (0.30)
SCHEMBL27553618 0.89 HTT (0.30)
SCHEMBL4101170 0.80 HTT (0.32)
SCHEMBL27756624 0.77 ALDH1A1 (0.40) TSHRCYP2C19GAA
SCHEMBL7718861 0.75 ALDH1A1 (0.36)
SCHEMBL27573906 0.73
SCHEMBL27573913 0.73
SCHEMBL5874768 0.72 ALDH1A1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100383121-C Substituted benzyl ester and its preparation process and novel process for preparing substituted mopipe therefrom TIANJIN TAIPU PHARMACEUTICAL S (CN) 2008-04-23 CN disclosed
CN-1827598-A Substituted benzyl ester and its preparation process and novel process for preparing substituted mopipe therefrom TIANJIN TAIPU PHARMACEUTICAL S (CN) 2006-09-06 CN disclosed
US-6140502-A Heat-based process for the re-racemisation of a (-)-2-phenylmethyl-3,3-dimethyl-piperidin-4-on derivative BOEHRINGER INGELHEIM KG (DE) 2000-10-31 US disclosed
US-6136980-A Method of preparing norbenzomorphane as an intermediate in the preparation of pharmaceutically useful benzomorphane derivatives, in particular (-)-(1R,5S,2\"R)-3'-hydroxy-2-(2-methoxypropyl)-5,9,9-trimethyl-6,7-benzo morphane BOEHRINGER INGELHEIM KG (DE) 2000-10-24 US disclosed
US-6054604-A Method of preparing norbenzomorphane as an intermediate BOEHRINGER INGELHEIM KG (DE) 2000-04-25 US disclosed
US-5945535-A Method of preparing norbenzomorphanes BOEHRINGER INGELHEIM KG (DE) 1999-08-31 US disclosed