SCHEMBL8034177

SCHEMBL8034177

S=C1N=NC(c2ccsc2)=N1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 9/20 0.39
CYP2B6 P20813 3/20 0.39
CYP2E1 P05181 2/20 0.39
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CCNB2 O95067 1/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
GSK3B P49841 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
CCNB3 Q8WWL7 1/20 0.34
TDO2 P48775 1/20 0.33
CYP17A1 P05093 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
KCNH2 Q12809 1/20 0.33
PDGFRB P09619 4/20 0.32
PDGFRA P16234 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8042073 0.72 MAPT (0.43) CYP3A4CYP2C9CYP2C19
SCHEMBL8189927 0.72 CYP2A6 (0.43) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C9
SCHEMBL4877279 0.70 ALDH1A1 (0.38)
SCHEMBL2125063 0.67 CYP2A6 (0.72) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C9
SCHEMBL8183577 0.64 CYP2A6 (0.43) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C9
SCHEMBL9465032 0.63 CYP2A6 (0.42) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C9
SCHEMBL8044653 0.63 BACE1 (0.35) BACE1
SCHEMBL3500357 0.63 CYP2A6 (0.42) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C9
SCHEMBL8043972 0.62 ALDH1A1 (0.45) GSK3BTDO2
SCHEMBL8048177 0.62 RAB9A (0.37) PDGFRBPDGFRAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed