SCHEMBL8034894

SCHEMBL8034894

C=Cc1cc(C)cc(C)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 4/20 0.44
NOS3 P29474 2/20 0.44
NOS1 P29475 1/20 0.44
LMNA P02545 2/20 0.33
TP53 P04637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
POLB P06746 2/20 0.32
APOBEC3G Q9HC16 1/20 0.32
HSD17B10 Q99714 1/20 0.31
UHRF1 Q96T88 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KMT2A Q03164 2/20 0.30
MEN1 O00255 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MITF O75030 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
RAD52 P43351 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10816604 0.87 NOS2 (0.40) NOS2NOS3NOS1TP53TDP1
SCHEMBL9170444 0.79 TP53 (0.35) LMNATP53TDP1POLBAPOBEC3G
SCHEMBL9797794 0.79 NOS2 (0.40) NOS2NOS3NOS1KMT2AMEN1
SCHEMBL9797790 0.79 NOS2 (0.40) NOS2NOS3NOS1KMT2AMEN1
SCHEMBL1179474 0.77 NOS2 (0.34) NOS2TP53TDP1KMT2AMEN1
SCHEMBL29600243 0.76 NOS2 (0.44) NOS2NOS3NOS1LMNATP53
SCHEMBL29881992 0.76 KDM4E (0.36) NOS2NOS3NOS1LMNAPOLB
SCHEMBL9797864 0.76 KDM4E (0.36) NOS2NOS3NOS1LMNAPOLB
SCHEMBL3088815 0.76 NOS2 (0.44) NOS2NOS3NOS1LMNAPOLB
SCHEMBL1646533 0.76 NOS2 (0.44) NOS2NOS3NOS1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4680357-A ADHESIVES THE DOW CHEMICAL COMPANY (US) 1987-07-14 US claimed
US-3937764-A VINYL PYRIDINE-B-PROPIOLACTONE GRAFT POLYMERS DENKI ONKYO CO., LTD. (JA) 1976-02-10 US claimed
WO-2024092115-A2 MK2 INHIBITORS AND USES THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2024-05-02 WO disclosed
WO-2009106749-A2 DERIVATIVES OF N-HETEROCYCLIC-IMIDAZO[1,2-A]PYRIDINE-2-CARBOXAMIDES, PREPARATION THEREOF AND THERAPEUTIC APPLICATION THEREOF SANOFI-AVENTIS (FR) 2009-09-03 WO disclosed
EP-1585743-B1 2-(1H-INDAZOL-6-YLAMINO)- BENZAMIDE COMPOUNDS AS PROTEIN KINASES INHIBITORS USEFUL FOR THE TREATMENT OF OPHTHALMIC DISEASES PFIZER (US) 2007-05-23 EP disclosed
US-5543298-A ADDING SPECIFIED COMPOUND TO LIQUID SAMPLE, MEASURING RATE OF AUTOOXIDATION SPECTROPHOTOMETRICALLY OXIS INTERNATIONAL S.A. (FR) 1996-08-06 US disclosed
EP-0625209-B1 METHOD FOR ASSAYING THE SOD ACTIVITY BY USING A SELF- OXIDIZABLE COMPOUND NECESSARY FOR ITS IMPLEMENTATION, SELF- OXIDIZABLE COMPOUNDS AND PREPARATION THEREOF OXIS INT SA (FR) 1996-07-17 EP disclosed
EP-0625209-A1 METHOD FOR ASSAYING THE SOD ACTIVITY BY USING A SELF-OXIDIZABLE COMPOUND NECESSARY FOR ITS IMPLEMENTATION, SELF-OXIDIZABLE COMPOUNDS AND PREPARATION THEREOF. BIOXYTECH (FR) 1994-11-23 EP disclosed
WO-1993011258-A1 METHOD FOR ASSAYING THE SOD ACTIVITY BY USING A SELF-OXIDIZABLE COMPOUND NECESSARY FOR ITS IMPLEMENTATION, SELF-OXIDIZABLE COMPOUNDS AND PREPARATION THEREOF BIOXYTECH (FR) 1993-06-10 WO disclosed
EP-0137655-B1 RADIATION-SENSITIVE POLYMER COMPOSITION TORAY INDUSTRIES, INC. (JP) 1988-12-28 EP disclosed
US-4783391-A Radiation-sensitive polyamide polymer composition with anthraquinone monoazide TORAY INDUSTRIES, INC. (JP) 1988-11-08 US disclosed
EP-0119719-A1 Radiation sensitive polymer composition TORAY INDUSTRIES, INC. (JP) 1984-09-26 EP disclosed
US-4409343-A DIENE AND VINYLPHYRIDINE COPOLYMERS THE GENERAL TIRE & RUBBER COMPANY (US) 1983-10-11 US disclosed
US-4409290-A HEAT CURABLE ADHESIVE WHICH IS BLEND OF GRAFT COPOLYMER OF ACRYLIC MONOMER, AND VINYL PYRIDINE MONOMER WITH PHENOLIC RESIN THE GENERAL TIRE & RUBBER COMPANY (US) 1983-10-11 US disclosed
US-4355131-A Adhesion of rubber to glass fibers THE GENERAL TIRE & RUBBER COMPANY (US) 1982-10-19 US disclosed
US-4243743-A CARBOXYL-CONTAINING POLYAMIDE, UNSATURATED AMINE OR QUATERNARY AMMONIUM SALT TORAY INDUSTRIES, INC. (JP) 1981-01-06 US disclosed
US-4118439-A IONICALLY CROSSLINKED QUATERNARY AMMONIUM POLYMER RHONE-POULENC S.A. (FR) 1978-10-03 US disclosed
US-4016341-A REDUCING SCALE DEPOSITS BY COATING SURFACES WITH PHOSPHORIC ESTERS OR SALTS SHIN-ETSU CHEMICAL COMPANY LIMITED (JA) 1977-04-05 US disclosed
US-4006127-A Cationic diazacyanine dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1977-02-01 US disclosed
US-3937764-A VINYL PYRIDINE-B-PROPIOLACTONE GRAFT POLYMERS DENKI ONKYO CO., LTD. (JA) 1976-02-10 US disclosed