SCHEMBL8034971

SCHEMBL8034971

COCCCNC(=O)N(C)C(=O)c1cc(OCc2ccccc2)c(OC)cc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 4/20 0.44
MTNR1A P48039 3/20 0.44
SMPD1 P17405 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
APP P05067 4/20 0.40
KDM4E B2RXH2 3/20 0.40
LMNA P02545 3/20 0.40
NPC1 O15118 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CTSV O60911 1/20 0.39
CTSL P07711 1/20 0.39
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HTR1A P08908 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8034976 0.90 NPC1 (0.45) MTNR1BMTNR1ASMPD1HDAC1HDAC8
SCHEMBL8023140 0.88 MTNR1B (0.49) MTNR1BMTNR1ASMPD1HDAC1HDAC8
SCHEMBL8037073 0.86 APP (0.44) MTNR1BMTNR1ASMPD1HDAC1HDAC8
SCHEMBL8023145 0.84 KDM4E (0.45) SMPD1HDAC1HDAC8HDAC6APP
SCHEMBL8038358 0.82 HPGD (0.39) APPKDM4EALDH1A1HPGD
SCHEMBL8023147 0.82 APP (0.46) SMPD1HDAC1HDAC8HDAC6APP
SCHEMBL8039245 0.82 MRGPRX4 (0.49) MTNR1BMTNR1ASMPD1HDAC1HDAC8
SCHEMBL8039269 0.82 ALDH1A1 (0.43) SMPD1HDAC1HDAC8HDAC6APP
SCHEMBL8037077 0.79 MEN1 (0.42) SMPD1HDAC1HDAC8HDAC6APP
SCHEMBL8025476 0.79 SMPD1 (0.47) SMPD1HDAC1HDAC8HDAC6APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed