SCHEMBL8035656

SCHEMBL8035656

CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N[C@H](N)Cc1ccc(-c2ccc(C#N)nc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.47
CTSC P53634 2/20 0.42
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
NPC1 O15118 1/20 0.40
JAK2 O60674 1/20 0.39
USP30 Q70CQ3 2/20 0.39
VHL P40337 1/20 0.39
ACACB O00763 1/20 0.39
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CPT2 P23786 1/20 0.38
CPT1A P50416 1/20 0.38
UCHL1 P09936 1/20 0.38
MC4R P32245 1/20 0.37
MC5R P33032 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075088 0.91 VHL (0.49) GPR119CTSCMEN1KMT2AJAK2
SCHEMBL2075087 0.91 VHL (0.49) GPR119CTSCMEN1KMT2AJAK2
SCHEMBL12383351 0.91 CTSC (0.53) GPR119CTSC
SCHEMBL8031921 0.83 GPR119 (0.47) GPR119CTSCMEN1KMT2ANPC1
SCHEMBL8035777 0.82 MEN1 (0.50) MEN1KMT2ANPC1USP30LMNA
SCHEMBL7859719 0.82 MEN1 (0.44) MEN1KMT2ANPC1LMNANPSR1
SCHEMBL3660022 0.80 GPR119 (0.45) GPR119CTSCMEN1KMT2AUSP30
SCHEMBL8028420 0.80 CTSC (0.40) CTSCMEN1KMT2ANPC1USP30
SCHEMBL2075366 0.78 VHL (0.54) CTSCVHL
SCHEMBL2074295 0.77 CTSC (0.59) CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed