SCHEMBL8036843

SCHEMBL8036843

CCNc1nc(-c2ccc(Cl)cc2)nc(C(C)C)c1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 3/20 0.45
NR4A2 P43354 3/20 0.45
NPSR1 Q6W5P4 3/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
FABP3 P05413 1/20 0.43
FABP4 P15090 1/20 0.43
FABP5 Q01469 1/20 0.43
KDM4E B2RXH2 1/20 0.43
PDE10A Q9Y233 1/20 0.42
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
ADORA3 P0DMS8 4/20 0.40
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
CYP1A1 P04798 2/20 0.38
CYP1A2 P05177 2/20 0.38
SELPLG Q14242 1/20 0.38
CHRNA7 P36544 1/20 0.38
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8034522 0.86 NPSR1 (0.47) RXRANR4A2NPSR1HPGDTSHR
SCHEMBL8034289 0.83 RXRA (0.43) RXRANR4A2NPSR1HPGDTSHR
SCHEMBL4011470 0.81 FABP3 (0.45) RXRANR4A2NPSR1HPGDTSHR
SCHEMBL8040520 0.81 NPSR1 (0.43) RXRANR4A2NPSR1HPGDTSHR
SCHEMBL4008510 0.78 FABP3 (0.43) RXRANR4A2NPSR1HPGDTSHR
SCHEMBL4008885 0.76 FABP3 (0.41) NPSR1HPGDFABP3FABP4FABP5
SCHEMBL4014246 0.76 MEN1 (0.46) RXRANR4A2NPSR1HPGDTSHR
SCHEMBL8032359 0.76 FABP3 (0.43) RXRANR4A2NPSR1HPGDTSHR
SCHEMBL8035080 0.75 TSHR (0.47) RXRANR4A2NPSR1HPGDTSHR
SCHEMBL4015161 0.75 ATM (0.54) RXRANR4A2NPSR1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080242-A1 SUBSTITUTED 4-AMINOPYRIMIDINE-5-CARBOXYLIC ACID AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed