SCHEMBL8038501

SCHEMBL8038501

CO[PH](=O)OCc1ccc(Br)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.45
MAOB P27338 6/20 0.41
APP P05067 1/20 0.38
HTR2A P28223 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
KDM4E B2RXH2 4/20 0.37
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
MAOA P21397 2/20 0.36
SMPD1 P17405 1/20 0.36
GLA P06280 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016123 0.88 IDO1 (0.52) IDO1MAOBAPPHTR2ATAAR1
SCHEMBL5051394 0.83 IDO1 (0.44) IDO1MAOBAPPHTR2ATAAR1
SCHEMBL673604 0.80 TSHR (0.44) IDO1MAOBKDM4EMAPTALDH1A1
SCHEMBL4938371 0.76 IDO1 (0.48) IDO1MAOBAPPHTR2ATAAR1
SCHEMBL7761382 0.75 IDO1 (0.54) IDO1MAOBMAPTALDH1A1KMT2A
Butane SCHEMBL2802241 0.74 POLB (0.42) IDO1MAOBAPPRXRARXRB
SCHEMBL7197241 0.72 IDO1 (0.55) IDO1MAOBAPPTAAR1ALDH1A1
SCHEMBL1995347 0.72 IDO1 (0.58) IDO1MAOBAPPHTR2ATAAR1
SCHEMBL9849327 0.71 TRPA1 (0.39) IDO1ALDH1A1CA2CA9
SCHEMBL5432093 0.71 AGXT (0.52) IDO1MAOBTAAR1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043341-A PHOSPHONYLATING AGENTS FOR REGIOSELECTIVE AND REPRODUCIBLE CONVERSION OF PEPTIDES TO PHOSPHONIC ACID PRODRUGS ELI LILLY & CO. (US) 2000-03-28 US disclosed
EP-0906915-A1 Preparation of cyclic peptide antifungal agents ELI LILLY AND COMPANY (US) 1999-04-07 EP disclosed
WO-1999006062-A1 CYCLIC PEPTIDE ANTIFUNGAL AGENTS ELI LILLY AND COMPANY (US) 1999-02-11 WO disclosed