SCHEMBL8038875

SCHEMBL8038875

CCC(=O)C(=Cc1ccccc1)C(=O)CC

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.63
KMT2A Q03164 1/20 0.63
AKR1C3 P42330 1/20 0.52
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
HTT P42858 1/20 0.52
RECQL P46063 1/20 0.48
TP53 P04637 1/20 0.48
MTNR1A P48039 2/20 0.47
MTNR1B P49286 2/20 0.47
FBP1 P09467 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
NR1H4 Q96RI1 1/20 0.46
NR1I2 O75469 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
AKR1C1 Q04828 1/20 0.45
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028857 0.92 KMT2A (0.56) MEN1KMT2AAKR1C3CES2CES1
SCHEMBL8028859 0.92 KMT2A (0.56) MEN1KMT2AAKR1C3CES2CES1
SCHEMBL28224152 0.88 MEN1 (0.60) MEN1KMT2ANR1H4CYP2C9LMNA
SCHEMBL28461515 0.86 MEN1 (0.84) MEN1KMT2AHTTALDH1A1NR1H4
SCHEMBL5804949 0.85 CA1 (0.56) MEN1KMT2AHTTALDH1A1CYP3A4
SCHEMBL5807201 0.85 CA1 (0.56) MEN1KMT2AHTTALDH1A1CYP3A4
SCHEMBL27690788 0.83 KMT2A (0.64) MEN1KMT2AHTTALDH1A1NR1H4
SCHEMBL31352034 0.83 AKR1C3 (0.64) MEN1KMT2AAKR1C3CES2CES1
SCHEMBL10665879 0.83 MEN1 (0.59) MEN1KMT2AAKR1C3CES2CES1
SCHEMBL30752455 0.83 RECQL (0.55) MEN1KMT2AAKR1C3CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108358831-A A kind of polysubstituted carbazole derivates and preparation method thereof 山东师范大学 2018-08-03 CN claimed
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP claimed
CN-108358831-B Polysubstituted carbazole derivative and preparation method thereof 山东师范大学 2020-09-29 CN disclosed
CN-108358831-A A kind of polysubstituted carbazole derivates and preparation method thereof 山东师范大学 2018-08-03 CN disclosed
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP disclosed
US-4719245-A TRIMERIZATION CATALYST THE DOW CHEMICAL COMPANY (US) 1988-01-12 US disclosed
US-4703099-A CATALYTICALLY TRIMERIZING ISOCYANATES THE DOW CHEMICAL COMPANY (US) 1987-10-27 US disclosed
US-4632989-A KETENE AMINAL-OLEFIN REACTION PRODUCT AS CATALYSTS THE DOW CHEMICAL COMPANY (US) 1986-12-30 US disclosed
US-4536490-A REACTION PRODUCT OF KETENE-AMINAL AND UNSATURATED COMPOUND THE UPJOHN COMPANY (US) 1985-08-20 US disclosed