SCHEMBL8039299

SCHEMBL8039299

Cc1ccc(CN2CC3OC3C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.53
S1PR5 Q9H228 1/20 0.53
LMNA P02545 2/20 0.52
ALDH1A1 P00352 1/20 0.52
POLB P06746 1/20 0.52
GBA1 P04062 1/20 0.51
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
CXCR4 P61073 1/20 0.46
HRH3 Q9Y5N1 2/20 0.46
HRH4 Q9H3N8 1/20 0.46
TEAD1 P28347 1/20 0.44
HRH1 P35367 1/20 0.44
MAPK1 P28482 2/20 0.43
MAPT P10636 1/20 0.43
ACHE P22303 2/20 0.43
BACE1 P56817 2/20 0.43
BCHE P06276 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12383 0.83 ALDH1A1 (0.55) S1PR1S1PR5LMNAALDH1A1POLB
SCHEMBL3107774 0.82 ALDH1A1 (0.52) S1PR5ALDH1A1MEN1KMT2AHRH3
SCHEMBL17850378 0.81 S1PR1 (0.50) S1PR1S1PR5LMNAALDH1A1POLB
SCHEMBL13229557 0.81 S1PR5 (0.46) S1PR5MAPTACHEBACE1BCHE
SCHEMBL2432513 0.80 SMN1; SMN2 (0.58) ALDH1A1MAPT
SCHEMBL2114892 0.80 FUCA1 (0.58) S1PR1S1PR5ALDH1A1GBA1ACHE
SCHEMBL11337029 0.80 FUCA1 (0.58) S1PR1S1PR5ALDH1A1GBA1ACHE
SCHEMBL11337025 0.80 FUCA1 (0.58) S1PR1S1PR5ALDH1A1GBA1ACHE
SCHEMBL17285918 0.78 S1PR1 (0.54) S1PR1S1PR5LMNAALDH1A1POLB
SCHEMBL22254430 0.78 S1PR1 (0.54) S1PR1S1PR5LMNAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227476-B1 TRICYCLIC TRIAZOLIC COMPOUNDS ESTEVE LABOR DR (ES) 2011-09-07 EP disclosed
EP-2070933-A1 Tricyclic triazolic compounds Laboratorios del Dr. Esteve S.A. (ES) 2009-06-17 EP disclosed
WO-2009071657-A1 TRICYCLIC TRIAZOLIC COMPOUNDS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2009-06-11 WO disclosed