SCHEMBL3107774

SCHEMBL3107774

Clc1ccc(CN2CC3OC3C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 2/20 0.52
SIGMAR1 Q99720 1/20 0.50
S1PR5 Q9H228 1/20 0.47
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
DRD4 P21917 4/20 0.43
LSS P48449 1/20 0.43
TEAD1 P28347 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
GAA P10253 1/20 0.43
HRH4 Q9H3N8 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
BACE1 P56817 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8039299 0.82 S1PR1 (0.53) ALDH1A1S1PR5MEN1KMT2ATEAD1
SCHEMBL13229557 0.82 S1PR5 (0.46) KDM4ESIGMAR1S1PR5DRD4BCHE
SCHEMBL11337025 0.82 FUCA1 (0.58) ALDH1A1SIGMAR1S1PR5CYP1A2CYP3A4
SCHEMBL2114892 0.82 FUCA1 (0.58) ALDH1A1SIGMAR1S1PR5CYP1A2CYP3A4
SCHEMBL11337029 0.82 FUCA1 (0.58) ALDH1A1SIGMAR1S1PR5CYP1A2CYP3A4
SCHEMBL2432513 0.78 SMN1; SMN2 (0.58) ALDH1A1KDM4ESIGMAR1DRD4MAPT
SCHEMBL2918814 0.78 ALDH1A1 (0.53) ALDH1A1KDM4ESIGMAR1S1PR5MEN1
SCHEMBL22731735 0.78 ALDH1A1 (0.53) ALDH1A1KDM4ESIGMAR1S1PR5MEN1
SCHEMBL2915354 0.78 ALDH1A1 (0.53) ALDH1A1KDM4ESIGMAR1S1PR5MEN1
SCHEMBL3771769 0.74 ALDH1A1 (0.50) ALDH1A1KDM4ESIGMAR1S1PR5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8399455-B2 Compounds useful as chemokine receptor antagonists MILLENNIUM PHARMACEUTICALS, INC. (US) 2013-03-19 US disclosed
US-20100234356-A1 COMPOUNDS USEFUL AS CHEMOKINE RECEPTOR ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-09-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100234356-A1 COMPOUNDS USEFUL AS CHEMOKINE RECEPTOR ANTAGONISTS ACKR3, CCR5, CXCR2 ALDH1A1 1889/4885KDM4E 4629/4885SIGMAR1 700/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.