SCHEMBL8039532

SCHEMBL8039532

CCOC(=O)/C=C/c1ccc(-n2cnc(C)c2)c(O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 2/20 0.60
DPP4 P27487 1/20 0.60
CYP3A4 P08684 1/20 0.54
MAOB P27338 1/20 0.52
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
APP P05067 7/20 0.48
FDPS P14324 1/20 0.47
PSEN1 P49768 2/20 0.47
PSEN2 P49810 2/20 0.47
APH1B Q8WW43 2/20 0.47
NCSTN Q92542 2/20 0.47
APH1A Q96BI3 2/20 0.47
PSENEN Q9NZ42 2/20 0.47
KCNH2 Q12809 1/20 0.45
IDO1 P14902 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12860064 0.90 TTR (0.51) TTRDPP4CYP3A4MAOBCA12
SCHEMBL1239568 0.87 PSEN1 (0.61) MAOBAPPFDPSPSEN1PSEN2
SCHEMBL1239565 0.87 PSEN1 (0.61) MAOBAPPFDPSPSEN1PSEN2
SCHEMBL8060709 0.78 KDM4E (0.43) APPPSEN1PSEN2APH1BNCSTN
SCHEMBL1239462 0.77 PSEN1 (0.54) APPPSEN1PSEN2APH1BNCSTN
SCHEMBL10281385 0.77 PSEN1 (0.40) APPPSEN1PSEN2APH1BNCSTN
Ethyl Caffeate SCHEMBL31059266 0.76 TTR (1.00) TTRDPP4CYP3A4MAOBCA12
Ethyl Caffeate SCHEMBL30286241 0.76 TTR (1.00) TTRDPP4CYP3A4MAOBCA12
Ethyl Caffeate SCHEMBL782033 0.76 TTR (1.00) TTRDPP4CYP3A4MAOBCA12
Ethyl Caffeate SCHEMBL22196845 0.76 TTR (1.00) TTRDPP4CYP3A4MAOBCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108766-A1 GAMMA SECRETASE MODULATORS FOR THE TREATMENT OF ALZHEIMER ' S DISEASE SCHERING CORPORATION (US) 2009-09-03 WO disclosed