SCHEMBL8040079

SCHEMBL8040079

Oc1ccc2sc(-c3ccccn3)nc2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.66
RAB9A P51151 5/20 0.66
NPC1 O15118 4/20 0.66
ALDH1A1 P00352 4/20 0.66
SMN1; SMN2 Q16637 3/20 0.66
TP53 P04637 2/20 0.66
HSD17B10 Q99714 2/20 0.66
TSHR P16473 1/20 0.66
MAPT P10636 3/20 0.55
NPSR1 Q6W5P4 1/20 0.55
APP P05067 2/20 0.50
MIF P14174 1/20 0.50
GABRA1 P14867 1/20 0.50
CBFB Q13951 1/20 0.48
LMNA P02545 2/20 0.48
POLB P06746 1/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
GAA P10253 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23954341 0.85 KDM4E (0.77) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL2949193 0.81 MIF (0.70) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL29081219 0.81 KDM4E (0.66) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL3207351 0.81 NPC1 (0.66) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL221431 0.80 NPC1 (1.00) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL2914054 0.79 APP (0.66) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL3202055 0.79 NPC1 (0.57) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL8050339 0.78 RAB9A (0.60) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL3201513 0.76 KDM4E (0.54) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL8358031 0.75 KDM4E (0.53) KDM4ERAB9ANPC1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed